SCHEMBL3720519

SCHEMBL3720519

O=C(NO)c1cc(-c2ccc(C#Cc3ccc(CN4CCOCC4)cc3)cc2)nc(NC(=O)C2CC2)n1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 3/20 0.52
TYK2 P29597 2/20 0.52
JAK2 O60674 1/20 0.52
JAK3 P52333 1/20 0.52
MMP13 P45452 7/20 0.50
MMP2 P08253 6/20 0.50
MMP8 P22894 6/20 0.50
MMP9 P14780 5/20 0.47
GSK3B P49841 1/20 0.46
DYRK1A Q13627 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13188455 0.94 JAK1 (0.56) JAK1TYK2JAK2JAK3GSK3B
SCHEMBL3714493 0.89 JAK1 (0.53) JAK1TYK2JAK2JAK3MMP13
SCHEMBL3718122 0.89 MOK (0.48) MMP13MMP2MMP8MMP9
SCHEMBL3710064 0.87 KDM4E (0.48) MMP13MMP2MMP8MMP9
SCHEMBL3714015 0.86 JAK2 (0.44) JAK2JAK3MMP13MMP2MMP8
SCHEMBL13187726 0.85 ALK (0.45) MMP13MMP2MMP8
SCHEMBL3713257 0.84 MMP2 (0.42) JAK2JAK3MMP13MMP2MMP8
SCHEMBL3716618 0.83 MMP2 (0.48) MMP13MMP2MMP8MMP9
SCHEMBL13187912 0.82 HDAC1 (0.41) JAK2JAK3MMP13MMP2MMP8
SCHEMBL13188579 0.81 HDAC1 (0.42) MMP13MMP2MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed