SCHEMBL3720675

SCHEMBL3720675

CC(=O)NCCc1ccc2nc(Oc3ccc(NC(C)C)cc3C)ccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.50
MTNR1B P49286 2/20 0.50
POLB P06746 1/20 0.38
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
PTGS1 P23219 1/20 0.37
BLM P54132 1/20 0.37
HIF1A Q16665 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PKM P14618 1/20 0.37
CES2 O00748 1/20 0.36
PIM1 P11309 2/20 0.36
RAF1 P04049 1/20 0.36
CSNK2A1 P68400 1/20 0.35
SCN9A Q15858 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718309 0.90 MTNR1A (0.49) MTNR1AMTNR1BMAPTKDM4EALDH1A1
SCHEMBL3717456 0.85 MTNR1A (0.50) MTNR1AMTNR1BMAPTKDM4EALDH1A1
SCHEMBL3719941 0.84 MTNR1A (0.51) MTNR1AMTNR1BMAPTKDM4EALDH1A1
SCHEMBL3721521 0.83 MTNR1A (0.48) MTNR1AMTNR1BPKMCES2SCN9A
SCHEMBL3727352 0.81 MTNR1A (0.50) MTNR1AMTNR1BMAPTKDM4EALDH1A1
SCHEMBL3726805 0.80 MTNR1A (0.49) MTNR1AMTNR1BMAPTKDM4EALDH1A1
SCHEMBL3720672 0.80 ACACB (0.38)
SCHEMBL3727615 0.80 MTNR1A (0.48) MTNR1AMTNR1BMAPTKDM4EALDH1A1
SCHEMBL3720627 0.79 MTNR1A (0.50) MTNR1AMTNR1BMAPTKDM4EALDH1A1
SCHEMBL3720171 0.79 MTNR1A (0.57) MTNR1AMTNR1BPOLBMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed