SCHEMBL3719941

SCHEMBL3719941

CC(=O)NCCc1ccc2nc(Oc3cccc(NC(C)C)c3)ccc2c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.51
MTNR1B P49286 5/20 0.51
ACACB O00763 2/20 0.43
CES2 O00748 1/20 0.41
SCN9A Q15858 2/20 0.41
GLI1 P08151 1/20 0.39
GLI2 P10070 1/20 0.39
RAF1 P04049 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
PTGS1 P23219 1/20 0.38
BLM P54132 1/20 0.38
HIF1A Q16665 1/20 0.38
HSD17B10 Q99714 1/20 0.38
RAD52 P43351 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722736 0.84 TAAR1 (0.36) SCN9A
SCHEMBL3720675 0.84 MTNR1A (0.50) MTNR1AMTNR1BCES2SCN9ARAF1
SCHEMBL3718309 0.83 MTNR1A (0.49) MTNR1AMTNR1BCES2KDM4EALDH1A1
SCHEMBL3722768 0.82 MTNR1A (0.50) MTNR1AMTNR1BACACBSCN9ASMN1; SMN2
SCHEMBL3720171 0.82 MTNR1A (0.57) MTNR1AMTNR1BACACBSCN9ARAF1
SCHEMBL3723899 0.82 KCNH3 (0.36) SCN9AALDH1A1MAPT
SCHEMBL3724455 0.81 KCNH3 (0.37) SCN9A
SCHEMBL3727055 0.81 ACACB (0.56) MTNR1AMTNR1BACACBSCN9ASMN1; SMN2
SCHEMBL3723898 0.81 PDE4B (0.50) SMN1; SMN2LMNAMAPT
SCHEMBL3726202 0.79 ACACB (0.58) MTNR1AMTNR1BACACBSCN9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed