SCHEMBL3721089

SCHEMBL3721089

CC(=O)c1ccc2nc(Oc3ccc(OC(C)C)c(C)c3)ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.53
ALDH1A1 P00352 5/20 0.41
TSHR P16473 2/20 0.41
SCN7A Q01118 1/20 0.38
KCNH2 Q12809 1/20 0.38
SCN9A Q15858 1/20 0.38
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
MEN1 O00255 1/20 0.37
PKM P14618 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 2/20 0.37
ESRRA P11474 1/20 0.35
CYP2A6 P11509 1/20 0.35
PPARG P37231 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GAA P10253 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
BCHE P06276 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721868 0.92 PDE4B (0.48) PDE4BALDH1A1TSHRSCN7AKCNH2
SCHEMBL3716835 0.89 PDE4B (0.53) PDE4BALDH1A1TSHRSCN7AKCNH2
SCHEMBL3720788 0.88 PDE4B (0.52) PDE4BALDH1A1TSHRSCN7AKCNH2
SCHEMBL3724294 0.86 PDE4B (0.55) PDE4BALDH1A1TSHRSCN7AKCNH2
SCHEMBL3719669 0.85 PDE4B (0.49) PDE4BALDH1A1TSHRSCN7AKCNH2
SCHEMBL3717722 0.85 PDE4B (0.45) PDE4BALDH1A1TSHRSCN7AKCNH2
SCHEMBL3719225 0.84 PDE4B (0.46) PDE4BALDH1A1TSHRSCN7AKCNH2
SCHEMBL3720702 0.82 PDE4B (0.57) PDE4BALDH1A1TSHRSCN7AKCNH2
SCHEMBL3717769 0.82 PDE4B (0.48) PDE4BALDH1A1HPGDMEN1KMT2A
SCHEMBL3719548 0.82 PDE4B (0.48) PDE4BALDH1A1TSHRSCN7AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed