SCHEMBL3720702

SCHEMBL3720702

CC(=O)c1ccc2nc(Oc3ccc(O)c(C)c3)ccc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.57
ESRRA P11474 2/20 0.44
SCN9A Q15858 2/20 0.41
SCN7A Q01118 2/20 0.41
KCNH2 Q12809 2/20 0.41
CYP2A6 P11509 1/20 0.39
PPARG P37231 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
BCHE P06276 2/20 0.38
ACHE P22303 2/20 0.38
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GLA P06280 1/20 0.36
SCN5A Q14524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721089 0.82 PDE4B (0.53) PDE4BESRRASCN9ASCN7AKCNH2
SCHEMBL3717735 0.81 PDE4B (0.57) PDE4BSCN9ASCN7AKCNH2CYP2A6
SCHEMBL3720071 0.79 PDE4B (0.49) PDE4BESRRASCN9ASCN7AKCNH2
SCHEMBL3717034 0.79 SCN7A (0.49) PDE4BSCN7AKCNH2PPARGSMN1; SMN2
SCHEMBL3720433 0.79 SCN7A (0.49) PDE4BSCN7AKCNH2PPARGSMN1; SMN2
SCHEMBL3721868 0.79 PDE4B (0.48) PDE4BSCN9ASCN7AKCNH2CYP2A6
SCHEMBL28248095 0.79 NPC1 (0.44) ESRRASMN1; SMN2GAATSHRNPSR1
SCHEMBL3724294 0.79 PDE4B (0.55) PDE4BSCN9ASCN7AKCNH2SMN1; SMN2
SCHEMBL3720703 0.78 PDE4B (0.36) PDE4BESRRASCN9ASCN7AKCNH2
SCHEMBL3718481 0.78 PDE4B (0.54) PDE4BSCN9APPARGSMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed