SCHEMBL3719669

SCHEMBL3719669

CC(=O)c1ccc2nc(Oc3ccc(OC(C)C4CC4)cc3C)ccc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.49
SCN9A Q15858 3/20 0.38
SCN7A Q01118 1/20 0.38
KCNH2 Q12809 1/20 0.38
ALDH1A1 P00352 3/20 0.34
TSHR P16473 1/20 0.34
KDM2B Q8NHM5 1/20 0.34
MAPK14 Q16539 1/20 0.34
BCHE P06276 2/20 0.33
ACHE P22303 2/20 0.33
HSF1 Q00613 1/20 0.33
PPARG P37231 1/20 0.33
ALOX5 P09917 1/20 0.33
GRM1 Q13255 1/20 0.33
MEN1 O00255 1/20 0.33
PKM P14618 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP2A6 P11509 1/20 0.33
ACACB O00763 1/20 0.33
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721868 0.91 PDE4B (0.48) PDE4BSCN9ASCN7AKCNH2ALDH1A1
SCHEMBL3721089 0.85 PDE4B (0.53) PDE4BSCN9ASCN7AKCNH2ALDH1A1
SCHEMBL3719225 0.84 PDE4B (0.46) PDE4BSCN9ASCN7AKCNH2ALDH1A1
SCHEMBL3726370 0.84 PDE4B (0.47) PDE4BSCN9ASCN7AKCNH2ALDH1A1
SCHEMBL3720793 0.84 ACACB (0.46) ACACB
SCHEMBL3724232 0.83 PDE4B (0.46) PDE4BALDH1A1KDM2BPPARGACACB
SCHEMBL3724295 0.82 PDE4B (0.46) PDE4BALDH1A1TSHRPPARGPKM
SCHEMBL3721926 0.81 PDE4B (0.44) PDE4BKDM2BACACB
SCHEMBL3720071 0.80 PDE4B (0.49) PDE4BSCN9ASCN7AKCNH2MAPK14
SCHEMBL3717291 0.80 MAPT (0.34) PDE4BSCN9AALDH1A1TSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed