SCHEMBL3721095

SCHEMBL3721095

COc1nc(CN)cc(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.49
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
MEN1 O00255 2/20 0.44
TSHR P16473 2/20 0.44
KMT2A Q03164 2/20 0.44
ATM Q13315 2/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 2/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
ACP1 P24666 3/20 0.40
PPARD Q03181 2/20 0.40
MAPK1 P28482 2/20 0.40
RAB9A P51151 1/20 0.40
F2RL3 Q96RI0 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3717005 0.86 CTSS (0.47) CTSSCTSKATMMAPTIDO1
SCHEMBL3728870 0.85 CTSS (0.42) CTSSCTSKIDO1TDO2PPARD
SCHEMBL3717780 0.83 CTSS (0.42) CTSSCTSKIDO1TDO2PPARD
SCHEMBL3725421 0.82 DPP4 (0.50) HSD17B10CTSSCTSKKDM4EPPARD
SCHEMBL3727413 0.81 CTSS (0.49) CTSSCTSKPPARDADORA3LTA4H
SCHEMBL3724728 0.80 KDM4E (0.49) HSD17B10CTSSCTSKKDM4EALDH1A1
SCHEMBL3717919 0.80 CTSS (0.47) CTSSCTSKKDM4EPPARDADORA3
SCHEMBL3724702 0.79 CTSS (0.47) CTSSCTSKMAPTPPARDALDH1A1
SCHEMBL3720125 0.78 CTSS (0.46) CTSSCTSKMEN1KMT2AMAPT
SCHEMBL3721220 0.77 KIF11 (0.51) CTSSCTSKPPARDRAB9AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US claimed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO claimed
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed