SCHEMBL3721766

SCHEMBL3721766

Cc1cccc(-n2nnc(CCSc3nnc(-c4cc[nH]c(=O)c4)n3C)n2)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.48
DRD2 P14416 9/20 0.45
DRD3 P35462 8/20 0.45
KCNH2 Q12809 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
DRD4 P21917 1/20 0.42
LMNA P02545 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
TP53 P04637 2/20 0.38
NPC1 O15118 1/20 0.38
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724363 0.84 DRD2 (0.43) GRM5DRD2DRD3KCNH2NPSR1
SCHEMBL3726056 0.80 GRM5 (0.57) GRM5DRD2NPSR1LMNAALDH1A1
SCHEMBL3110804 0.79 GRM5 (0.59) GRM5DRD2DRD3KCNH2NPSR1
SCHEMBL3110795 0.79 GRM5 (0.59) GRM5DRD2DRD3KCNH2NPSR1
SCHEMBL3722888 0.78 GRM5 (0.48) GRM5DRD2DRD3KCNH2NPSR1
SCHEMBL18490899 0.74 NPC1 (0.61) DRD2DRD3KCNH2CHRM1CHRM3
SCHEMBL17712859 0.73 DRD2 (0.54) DRD2DRD3KCNH2CHRM1CHRM3
SCHEMBL5479011 0.72 KMT2A (0.44) GRM5LMNAALDH1A1NPC1MEN1
SCHEMBL2897521 0.71 ALOX12 (0.56) DRD2DRD3NPSR1LMNAALDH1A1
SCHEMBL5741042 0.67 MAPT (0.51) LMNAALDH1A1RXFP1NPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010123451-A1 SULPHIDE BRIDGED DERIVATIVES AS MODULATORS OF MGLUR5 ASTRAZENECA AB (SE) 2010-10-28 WO claimed