SCHEMBL3722347

SCHEMBL3722347

CC(NC(=O)C1(NC(=O)Oc2cncnc2)CC1)c1ccc(Oc2ccc(Br)cc2C(F)(F)F)cn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 4/20 0.36
CACNA1G O43497 2/20 0.36
CACNA1H O95180 2/20 0.36
CNR2 P34972 1/20 0.36
KCNH2 Q12809 1/20 0.36
BDKRB1 P46663 10/20 0.35
CNR1 P21554 3/20 0.32
FAAH O00519 2/20 0.32
TRPV1 Q8NER1 2/20 0.32
PSMB11 A5LHX3 1/20 0.31
PSMA7 O14818 1/20 0.31
PSMB1 P20618 1/20 0.31
PSMA1 P25786 1/20 0.31
PSMA2 P25787 1/20 0.31
PSMA3 P25788 1/20 0.31
PSMA4 P25789 1/20 0.31
PSMB8 P28062 1/20 0.31
PSMB9 P28065 1/20 0.31
PSMA5 P28066 1/20 0.31
PSMB4 P28070 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722282 0.91 CACNA1I (0.38) CACNA1ICACNA1GCACNA1HCNR2KCNH2
SCHEMBL13191642 0.91 BDKRB1 (0.45) CACNA1ICACNA1GCACNA1HCNR2KCNH2
SCHEMBL3722571 0.91 CACNA1I (0.36) CACNA1ICACNA1GCACNA1HCNR2KCNH2
SCHEMBL14856578 0.86 BDKRB1 (0.34) CACNA1ICACNA1GCACNA1HCNR2KCNH2
SCHEMBL3725902 0.85 CACNA1I (0.37) CACNA1ICACNA1GCACNA1HBDKRB1CNR1
SCHEMBL3722413 0.85 CACNA1I (0.37) CACNA1ICACNA1GCACNA1HBDKRB1CNR1
SCHEMBL3729328 0.83 BDKRB1 (0.36) BDKRB1CNR1FAAHTRPV1
SCHEMBL13191405 0.83 BDKRB1 (0.45) CACNA1ICACNA1GCACNA1HCNR2KCNH2
SCHEMBL13191277 0.83 BDKRB1 (0.45) CACNA1ICACNA1GCACNA1HCNR2KCNH2
SCHEMBL13191728 0.82 BDKRB1 (0.45) CACNA1ICACNA1GCACNA1HCNR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed