SCHEMBL3725902

SCHEMBL3725902

COc1ccc(Oc2ccc([C@@H](C)NC(=O)C3(NC(=O)Oc4cncnc4)CC3)nc2)c(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 2/20 0.37
BDKRB1 P46663 4/20 0.37
CNR1 P21554 2/20 0.35
HPGDS O60760 2/20 0.35
FAAH O00519 3/20 0.34
TRPV1 Q8NER1 2/20 0.34
ACACB O00763 1/20 0.34
VNN1 O95497 3/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CACNA1G O43497 1/20 0.31
CACNA1H O95180 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722413 1.00 CACNA1I (0.37) CACNA1IBDKRB1CNR1HPGDSFAAH
SCHEMBL13191245 0.91 BDKRB1 (0.47) CACNA1IBDKRB1CNR1HPGDSACACB
SCHEMBL13191284 0.91 BDKRB1 (0.47) CACNA1IBDKRB1CNR1HPGDSACACB
SCHEMBL3722282 0.90 CACNA1I (0.38) CACNA1IBDKRB1CNR1HPGDSFAAH
SCHEMBL3723568 0.89 VNN1 (0.38) CACNA1IBDKRB1CNR1HPGDSACACB
SCHEMBL3722347 0.85 CACNA1I (0.36) CACNA1IBDKRB1CNR1FAAHTRPV1
SCHEMBL3722571 0.83 CACNA1I (0.36) CACNA1IBDKRB1CNR1CACNA1GCACNA1H
SCHEMBL13191288 0.82 BDKRB1 (0.47) CACNA1IBDKRB1CNR1HPGDSACACB
SCHEMBL3729328 0.81 BDKRB1 (0.36) BDKRB1CNR1FAAHTRPV1
SCHEMBL3722080 0.80 VNN1 (0.33) FAAHTRPV1VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed