SCHEMBL3729328

SCHEMBL3729328

COc1ccc(Oc2cnc(C(C)NC(=O)C3(NC(=O)Oc4cncnc4)CC3)nc2)c(C(F)(F)F)c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 13/20 0.36
CNR1 P21554 2/20 0.36
LIMK1 P53667 2/20 0.33
LIMK2 P53671 1/20 0.33
FAAH O00519 2/20 0.33
TRPV1 Q8NER1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722282 0.92 CACNA1I (0.38) BDKRB1CNR1LIMK1LIMK2FAAH
SCHEMBL13191628 0.91 BDKRB1 (0.45) BDKRB1CNR1
SCHEMBL13191246 0.85 BDKRB1 (0.37) BDKRB1
SCHEMBL3722571 0.84 CACNA1I (0.36) BDKRB1CNR1
SCHEMBL3722347 0.83 CACNA1I (0.36) BDKRB1CNR1FAAHTRPV1
SCHEMBL13191405 0.83 BDKRB1 (0.45) BDKRB1CNR1LIMK1
SCHEMBL3722860 0.83 GAA (0.33) LIMK1LIMK2FAAHTRPV1
SCHEMBL3722367 0.82 BDKRB1 (0.46) BDKRB1CNR1
SCHEMBL3718987 0.81 LIMK1 (0.37) LIMK1LIMK2
SCHEMBL3722413 0.81 CACNA1I (0.37) BDKRB1CNR1FAAHTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed