SCHEMBL3722973

SCHEMBL3722973

CCN(C(=O)OC(C)(C)C)c1nc(Cl)cc(N2CCOCC2)n1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
PIK3CA P42336 1/20 0.41
RAF1 P04049 1/20 0.40
BRAF P15056 1/20 0.40
AKT1 P31749 5/20 0.39
NAPEPLD Q6IQ20 6/20 0.37
GAA P10253 1/20 0.37
ATR Q13535 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722970 0.74 AKT1 (0.51) KMT2ACYP1A2CYP2D6MAPTRAF1
SCHEMBL29023026 0.72 GPR119 (0.47) MAPT
SCHEMBL16094927 0.72 CYP1A2 (0.60) KMT2ACYP1A2CYP2D6MAPTRAF1
SCHEMBL23505799 0.72 CYP1A2 (0.54) KMT2ACYP1A2CYP2D6MAPTRAF1
SCHEMBL18153347 0.72 PIK3CA (0.53) KMT2ACYP1A2CYP2D6MAPTPIK3CA
SCHEMBL29434915 0.72 PIK3CA (0.53) KMT2ACYP1A2CYP2D6MAPTPIK3CA
SCHEMBL3997637 0.72 PIK3CA (0.53) KMT2ACYP1A2CYP2D6MAPTPIK3CA
SCHEMBL244726 0.71 PIK3CA (0.40) KMT2APIK3CAGAA
SCHEMBL3605038 0.71 USP2 (0.48) KMT2ACYP1A2CYP2D6MAPTPIK3CA
SCHEMBL3115454 0.70 PIK3CA (0.39) KMT2APIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2146981-A1 PHARMACEUTICAL COMPOUNDS F. Hoffmann-Roche AG (CH) 2010-01-27 EP disclosed
WO-2008125833-A1 PHARMACEUTICAL COMPOUNDS PIRAMED LIMITED (GB) 2008-10-23 WO disclosed