SCHEMBL3722970

SCHEMBL3722970

CC(C)(C)OC(=O)NCCc1nc(Cl)cc(N2CCOCC2)n1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.51
BRD4 O60885 2/20 0.45
KMT2A Q03164 2/20 0.44
MAPT P10636 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
RAF1 P04049 1/20 0.42
BRAF P15056 1/20 0.42
DRD2 P14416 6/20 0.40
STK17B O94768 1/20 0.40
STK17A Q9UEE5 1/20 0.40
LMNA P02545 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
SUV39H2 Q9H5I1 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PRKDC P78527 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13119749 0.89 AKT1 (0.51) AKT1BRD4KMT2AMAPTLMNA
SCHEMBL13119769 0.79 SMN1; SMN2 (0.43) AKT1KMT2AMAPTCYP1A2CYP2D6
SCHEMBL3603746 0.78 ATR (0.49) AKT1PRKDC
SCHEMBL2073168 0.77 KMT2A (0.51) KMT2AMAPTCYP1A2CYP2D6RAF1
SCHEMBL3610408 0.77 RECQL (0.47) KMT2AMAPTLMNAKDM4EMEN1
SCHEMBL3988105 0.77 ALDH1A1 (0.53) AKT1BRD4MAPTSTK17BSTK17A
SCHEMBL24312197 0.76 AKT1 (0.43) AKT1BRD4KMT2AMAPTCYP1A2
SCHEMBL3722973 0.74 KMT2A (0.44) AKT1KMT2AMAPTCYP1A2CYP2D6
SCHEMBL3605615 0.74 KCNK3 (0.43) AKT1KMT2AMAPTCYP1A2CYP2D6
SCHEMBL13142298 0.74 KCNK3 (0.43) AKT1KMT2AMAPTCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2146981-A1 PHARMACEUTICAL COMPOUNDS F. Hoffmann-Roche AG (CH) 2010-01-27 EP disclosed
WO-2008125833-A1 PHARMACEUTICAL COMPOUNDS PIRAMED LIMITED (GB) 2008-10-23 WO disclosed
WO-2008125833-A1 PHARMACEUTICAL COMPOUNDS PIRAMED LIMITED (GB) 2008-10-23 WO disclosed