SCHEMBL3723394

SCHEMBL3723394

CN1CCC(Nc2cc(Cl)cc3cc(-c4ccccc4)[nH]c23)CC1.Clc1cc(NC2CCN(Cc3ccccc3)C2)c2[nH]c(-c3ccccc3)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.44
ACHE P22303 3/20 0.44
BACE1 P56817 3/20 0.44
ROCK2 O75116 4/20 0.44
CCR2 P41597 3/20 0.44
ROCK1 Q13464 3/20 0.44
DRD2 P14416 2/20 0.42
DRD4 P21917 2/20 0.42
EHMT2 Q96KQ7 2/20 0.42
KAT2B Q92831 3/20 0.42
ITK Q08881 1/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
ADORA2B P29275 1/20 0.41
CNR1 P21554 1/20 0.41
OPRK1 P41145 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3003745 0.94 BCHE (0.49) BCHEACHEBACE1ROCK2CCR2
SCHEMBL3009562 0.89 VCP (0.43) KAT2BKDM4E
SCHEMBL3415042 0.78 VCP (0.48)
SCHEMBL3003738 0.78 VCP (0.44) ITK
SCHEMBL3008763 0.78 POLB (0.50) ITK
SCHEMBL3432708 0.78 MAPK8 (0.48) CNR1
SCHEMBL3005194 0.78 ADORA1 (0.45) KDM4EGAA
SCHEMBL29205628 0.77 VCP (0.40) EHMT2GAA
SCHEMBL30182989 0.77 VCP (0.40) EHMT2GAA
SCHEMBL3005392 0.77 NPC1 (0.41) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2178870-A1 INDOLE AND INDAZOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG Life Sciences Ltd. (KR) 2010-04-28 EP disclosed
WO-2009025478-A1 INDOLE AND INDAZOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG LIFE SCIENCES LTD. (KR) 2009-02-26 WO disclosed