SCHEMBL3724316

SCHEMBL3724316

C[C@H](CS(=O)(=O)c1ccc(OCC(F)(F)F)cc1Cl)C(=O)N1CCCC1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 8/20 0.41
REN P00797 4/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
F2 P00734 1/20 0.41
LTA4H P09960 1/20 0.41
MAPT P10636 1/20 0.41
PEPD P12955 1/20 0.41
ALOX15 P16050 1/20 0.41
PTGS1 P23219 1/20 0.41
HTR2A P28223 1/20 0.41
PTGS2 P35354 1/20 0.41
HRH1 P35367 1/20 0.41
THPO P40225 1/20 0.41
PMP22 Q01453 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ACE2 Q9BYF1 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ITGB1 P05556 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718279 0.88 ITGB1 (0.40) NPSR1ALDH1A1ITGB1ITGA4CTSS
SCHEMBL3716347 0.83 ACE (0.49) ACERENLMNAKDM4EF2
SCHEMBL3718797 0.79 ACE (0.51) ACERENLMNAKDM4EF2
SCHEMBL3723409 0.76 CTSS (0.41) NPSR1ALDH1A1ITGB1ITGA4CTSS
SCHEMBL3065367 0.74 CTSS (0.51) CTSS
SCHEMBL3060617 0.71 CTSS (0.50) CTSS
SCHEMBL3718817 0.71 ACE (0.40) ACERENALDH1A1
SCHEMBL3065890 0.70 CTSS (0.52) CTSS
SCHEMBL24668844 0.69 ACE (0.52) ACERENLMNAKDM4EF2
SCHEMBL3067366 0.68 CTSS (0.53) ITGB1ITGA4CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed