SCHEMBL3723409

SCHEMBL3723409

O=C(O)C1CCCN1C(=O)c1ccc(S(=O)(=O)c2ccc(OCC(F)(F)F)cc2Cl)cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.41
SFRP1 Q8N474 4/20 0.40
WNT3 P56703 3/20 0.40
ALDH1A1 P00352 1/20 0.39
CA2 P00918 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
MCL1 Q07820 1/20 0.38
ITGB1 P05556 1/20 0.38
ITGA4 P13612 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
RORC P51449 1/20 0.37
HSD11B1 P28845 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724316 0.76 ACE (0.41) CTSSALDH1A1ITGB1ITGA4NPSR1
SCHEMBL3718279 0.74 ITGB1 (0.40) CTSSALDH1A1L3MBTL1ITGB1ITGA4
SCHEMBL3062005 0.73 CTSS (0.49) CTSSALDH1A1
SCHEMBL13146441 0.69 CCR2 (0.54) MCL1
SCHEMBL3723608 0.69 RORC (0.38) CTSSITGB1ITGA4RORCHSD11B1
SCHEMBL17313719 0.67 L3MBTL1 (0.42) SFRP1WNT3ALDH1A1CA2L3MBTL1
SCHEMBL14130046 0.67 HCRTR1 (0.39) ALDH1A1L3MBTL1NPSR1
SCHEMBL14130218 0.67 HCRTR1 (0.39) ALDH1A1L3MBTL1NPSR1
SCHEMBL3065890 0.66 CTSS (0.52) CTSS
SCHEMBL17428297 0.66 SCN9A (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed