SCHEMBL3724522

SCHEMBL3724522

Clc1cc2c(Cl)cc3c(Cl)cc(Cl)c4c(Cl)cc(c1Cl)c2c34

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.41
AHR P35869 15/20 0.41
HPGD P15428 3/20 0.36
HSD17B10 Q99714 3/20 0.36
TSHR P16473 2/20 0.36
CASP1 P29466 1/20 0.36
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3661470 0.87 AHR (0.38) CYP3A4AHRHPGDHSD17B10TSHR
SCHEMBL13000534 0.84 AHR (0.37) CYP3A4AHRHPGDHSD17B10TSHR
SCHEMBL29508980 0.79 CYP3A4 (0.53) CYP3A4AHRHPGDHSD17B10TSHR
SCHEMBL10311723 0.78 AHR (0.40) CYP3A4AHRHPGDHSD17B10TSHR
SCHEMBL28744259 0.74 CYP3A4 (0.53) CYP3A4AHRHPGDHSD17B10TSHR
SCHEMBL29857997 0.74 CYP3A4 (0.53) CYP3A4AHRHPGDHSD17B10TSHR
SCHEMBL29629138 0.74 CYP3A4 (0.53) CYP3A4AHRHPGDHSD17B10TSHR
SCHEMBL30681699 0.73 CYP3A4 (0.50) CYP3A4AHRHPGDHSD17B10TSHR
SCHEMBL10524296 0.73 AHR (0.41) CYP3A4AHRHPGDHSD17B10TSHR
SCHEMBL30485634 0.72 ALDH1A1 (0.55) CYP3A4AHRHPGDHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796456-B2 Naphthalene diimide compounds UNIVERSITY COLLEGE LONDON (GB) 2014-08-05 US disclosed
EP-2227470-B1 NAPHTHALENE DIIMIDE COMPOUNDS INTERACTING WITH G-QUADRPLEX REGIONS IN DNA UNIV LONDON (GB) 2014-03-05 EP disclosed
US-20100311739-A1 Naphthalene Diimide Compounds UNIVERSITY COLLEGE LONDON (GB) 2010-12-09 US disclosed
EP-2227470-A1 NAPHTHALENE DIIMIDE COMPOUNDS INTERACTING WITH G-QUADRUPLEX REGIONS IN DNA THE SCHOOL OF PHARMACY, UNIVERSITY OF LONDON (GB) 2010-09-15 EP disclosed
WO-2009068916-A1 NAPHTHALENE DIIMIDE COMPOUNDS INTERACTING WITH G-QUADRUPLEX REGIONS IN DNA SCHOOL OF PHARMACY, UNIVERSITY OF LONDON (GB) 2009-06-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100311739-A1 Naphthalene Diimide Compounds NDC1, NUTF2, NDUFC2 CYP3A4 821/4885AHR 127/4885HPGD 286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.