SCHEMBL3728344

SCHEMBL3728344

CCCCCc1ccnc2[nH]c3ccc(/C=C/c4ccc(OC)cc4)cc3c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 2/20 0.52
CCNB2 O95067 3/20 0.43
CDK1 P06493 3/20 0.43
CCNB1 P14635 3/20 0.43
GSK3A P49840 3/20 0.43
GSK3B P49841 3/20 0.43
CCNB3 Q8WWL7 3/20 0.43
GLA P06280 2/20 0.42
AHR P35869 1/20 0.42
GHSR Q92847 1/20 0.41
UTS2R Q9UKP6 2/20 0.40
CDK5 Q00535 2/20 0.40
CDK5R1 Q15078 2/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
ZAP70 P43403 1/20 0.40
PTK2B Q14289 1/20 0.40
PTK6 Q13882 2/20 0.39
NPC1 O15118 2/20 0.38
CYP1A2 P05177 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3728347 1.00 ALK (0.52) ALKCCNB2CDK1CCNB1GSK3A
SCHEMBL675009 0.90 ALK (0.50) ALKCCNB2CDK1CCNB1GSK3A
SCHEMBL3727396 0.88 ALK (0.47) ALKGLAUTS2RNPC1CYP1A2
SCHEMBL3727398 0.88 ALK (0.47) ALKGLAUTS2RNPC1CYP1A2
SCHEMBL3719653 0.86 ALK (0.54) ALKCCNB2CDK1CCNB1GSK3A
SCHEMBL3725131 0.82 ALK (0.47) ALKGHSRUTS2R
SCHEMBL675008 0.80 ALK (0.48) ALKCCNB2CDK1CCNB1GSK3A
SCHEMBL676373 0.80 ALK (0.76) ALKGLAPTK6NPC1CYP1A2
SCHEMBL675670 0.80 GHSR (0.40) ALKCCNB2CDK1CCNB1GSK3A
SCHEMBL3723526 0.79 TUBB4A (0.45) ALKCCNB2CDK1CCNB1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed