SCHEMBL3728859

SCHEMBL3728859

Cc1c(OCCN2CCOCC2)cccc1[N+](=O)[O-]

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.68
CYP1A2 P05177 1/20 0.68
CYP2C19 P33261 1/20 0.68
SMN1; SMN2 Q16637 4/20 0.58
KDM4E B2RXH2 5/20 0.55
ALDH1A1 P00352 4/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
POLB P06746 2/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
LTA4H P09960 1/20 0.50
PTGS1 P23219 1/20 0.50
PTGS2 P35354 1/20 0.50
TDP1 Q9NUW8 1/20 0.48
DRD1 P21728 1/20 0.48
DRD4 P21917 1/20 0.48
DRD5 P21918 1/20 0.48
TSHR P16473 1/20 0.47
P2RY12 Q9H244 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14453656 0.89 LTA4H (0.62) CYP2D6CYP1A2CYP2C19KDM4EALDH1A1
SCHEMBL1852361 0.87 CYP2D6 (0.88) CYP2D6CYP1A2CYP2C19SMN1; SMN2KDM4E
SCHEMBL2029093 0.85 CYP1A2 (0.68) CYP2D6CYP1A2CYP2C19SMN1; SMN2KDM4E
SCHEMBL216475 0.85 CYP1A2 (0.68) CYP2D6CYP1A2CYP2C19SMN1; SMN2KDM4E
SCHEMBL25378553 0.85 CYP1A2 (0.68) CYP2D6CYP1A2CYP2C19SMN1; SMN2KDM4E
SCHEMBL5237000 0.83 CYP1A2 (0.65) CYP2D6CYP1A2CYP2C19SMN1; SMN2KDM4E
SCHEMBL5239956 0.82 CYP2D6 (0.64) CYP2D6CYP1A2CYP2C19SMN1; SMN2KDM4E
SCHEMBL13744516 0.79 SMN1; SMN2 (0.66) CYP2D6SMN1; SMN2KDM4EALDH1A1POLB
SCHEMBL28937449 0.78 POLB (0.64) CYP2D6SMN1; SMN2KDM4EALDH1A1POLB
SCHEMBL3725632 0.78 SMN1; SMN2 (0.64) CYP2D6SMN1; SMN2KDM4EPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125103-A1 DIKETOPIPERAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LIMITED (GB) 2010-11-04 WO disclosed