SCHEMBL372927

SCHEMBL372927

BrCc1ccc(Oc2ccc[nH]2)cc1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
LTA4H P09960 1/20 0.33
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
ST14 Q9Y5Y6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL79800 0.76 LTA4H (0.50) TRPA1TSHRLTA4H
SCHEMBL5885219 0.75 ST14 (0.48) TRPA1ALDH1A1TSHRLTA4HCES2
SCHEMBL29171477 0.74 LTA4H (0.48) TRPA1TSHRLTA4H
SCHEMBL9651942 0.72 DAO (0.35)
SCHEMBL751190 0.71 LTA4H (0.61) TRPA1ALDH1A1TSHRLTA4HCES2
Dimethylamine SCHEMBL10731360 0.69 LTA4H (0.53) TRPA1ALDH1A1TSHRLTA4H
SCHEMBL182793 0.68
SCHEMBL28667800 0.67 HDAC1 (0.44) TRPA1ALDH1A1TSHRCES2CES1
SCHEMBL28914769 0.66 AURKA (0.36)
Hydrochloric Acid SCHEMBL6344142 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408756-A1 ALPHA-(N-BENZENESULFONAMIDO)CYCLOALKYL DERIVATIVES Bristol-Myers Squibb Company (US) 2012-01-25 EP disclosed
WO-2010108067-A1 ALPHA-(N-BENZENESULFONAMIDO)CYCLOALKYL DERIVATIVES BRISTOL-MYERS SQUIBB COMPANY (US) 2010-09-23 WO disclosed