SCHEMBL3739617

SCHEMBL3739617

COc1c(C#N)ccc(C2CCCC2)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.43
ALOX5AP P20292 6/20 0.40
FEN1 P39748 6/20 0.40
CHEK1 O14757 2/20 0.37
AR P10275 4/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
CEL P19835 2/20 0.34
PGR P06401 1/20 0.34
NR3C2 P08235 1/20 0.34
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3749818 0.98 HTR2A (0.42) HTR2AALOX5APFEN1CHEK1AR
SCHEMBL3747583 0.97 FEN1 (0.43) HTR2AALOX5APFEN1CHEK1AR
SCHEMBL3743094 0.94 HTR2A (0.39) HTR2AALOX5APFEN1CHEK1AR
SCHEMBL19614567 0.81 FEN1 (0.42) HTR2AALOX5APFEN1HCRTR1HCRTR2
SCHEMBL17729508 0.79 HTR2A (0.39) HTR2AALOX5APFEN1HCRTR1HCRTR2
SCHEMBL293119 0.79 KCNJ1 (0.36) HTR2AARPGR
SCHEMBL17202931 0.77 HTR2A (0.40) HTR2AALOX5APFEN1ARHCRTR1
SCHEMBL29058360 0.74 OPRL1 (0.40) HTR2AALOX5APFEN1HCRTR1HCRTR2
SCHEMBL2959996 0.70 KDM4E (0.44) ARPGRMAOAMAOB
SCHEMBL7961132 0.70 ALDH1A1 (0.48) ARPGRMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7834039-B2 Oxadiazole compounds ABBOTT LABORATORIES (US) 2010-11-16 US disclosed