SCHEMBL3740489

SCHEMBL3740489

NN(C(=O)C(c1ccccc1F)N1CCN2CCC[C@@H]2C1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.47
TACR1 P25103 17/20 0.41
MC4R P32245 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3667305 0.90 GHSR (0.47) GHSRTACR1
SCHEMBL3666028 0.90 GHSR (0.47) GHSRTACR1
SCHEMBL3634488 0.89 TACR1 (0.51) GHSRTACR1
SCHEMBL3666507 0.87 TACR1 (0.45) GHSRTACR1
SCHEMBL3801373 0.85 GHSR (0.50) GHSRTACR1
SCHEMBL3666109 0.85 GHSR (0.50) GHSRTACR1
SCHEMBL3724611 0.82 GHSR (0.69) GHSRTACR1
SCHEMBL3673888 0.82 GHSR (0.69) GHSRTACR1
SCHEMBL3636170 0.81 GHSR (0.42) GHSRTACR1
SCHEMBL3639324 0.80 GHSR (0.69) GHSRTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2167466-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR Glaxo Group Limited (GB) 2010-03-31 EP claimed
WO-2008148853-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2008-12-11 WO claimed
EP-2167466-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR Glaxo Group Limited (GB) 2010-03-31 EP disclosed
WO-2008148853-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2008-12-11 WO disclosed