SCHEMBL3747474

SCHEMBL3747474

CCc1nc(-c2ncccn2)sc1C(=O)NCc1ccc(OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.53
LMNA P02545 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
ALDH1A1 P00352 6/20 0.52
KMT2A Q03164 3/20 0.51
CYP1A2 P05177 3/20 0.51
CYP3A4 P08684 3/20 0.51
CYP2C9 P11712 3/20 0.51
CYP2C19 P33261 3/20 0.51
EGLN1 Q9GZT9 1/20 0.51
GAA P10253 1/20 0.51
MEN1 O00255 2/20 0.49
PPARA Q07869 1/20 0.48
RAB9A P51151 2/20 0.48
MAPT P10636 1/20 0.47
NPC1 O15118 1/20 0.47
CHRM4 P08173 1/20 0.47
KDM4E B2RXH2 1/20 0.46
POLB P06746 2/20 0.46
ATM Q13315 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3751769 0.89 EGLN1 (0.50) HPGDLMNASMN1; SMN2ALDH1A1KMT2A
SCHEMBL3743150 0.89 PPARA (0.55) HPGDSMN1; SMN2ALDH1A1CYP1A2CYP3A4
SCHEMBL3748773 0.88 EGLN1 (0.47) HPGDLMNASMN1; SMN2ALDH1A1KMT2A
SCHEMBL3749009 0.88 KMT2A (0.49) LMNAKMT2ACYP1A2CYP2C19PPARA
SCHEMBL3743433 0.85 MAOB (0.51) HPGDLMNASMN1; SMN2ALDH1A1KMT2A
SCHEMBL3743964 0.83 PTGDR2 (0.45) HPGDLMNASMN1; SMN2ALDH1A1KMT2A
SCHEMBL3747214 0.83 CHRM4 (0.46) CHRM4
SCHEMBL3748062 0.81 KCNA5 (0.47) HPGDLMNAKMT2ACYP3A4CYP2C9
SCHEMBL3738919 0.80 POLB (0.53) LMNAALDH1A1KMT2AMEN1POLB
SCHEMBL3738332 0.80 MAPK14 (0.53) HPGDKMT2AMEN1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9133204-B2 5-membered heterocyclic amides and related compounds H. LUNDBECK A/S (DK) 2015-09-15 US disclosed
US-9133204-B2 5-membered heterocyclic amides and related compounds H. LUNDBECK A/S (DK) 2015-09-15 US disclosed
US-9133204-B2 5-membered heterocyclic amides and related compounds H. LUNDBECK A/S (DK) 2015-09-15 US disclosed
EP-2178865-B1 5-MEMBERED HETEROCYCLIC AMIDES AND RELATED COMPOUNDS LUNDBECK H AS (DK) 2015-08-19 EP disclosed
EP-2178865-B1 5-MEMBERED HETEROCYCLIC AMIDES AND RELATED COMPOUNDS LUNDBECK H AS (DK) 2015-08-19 EP disclosed
US-20150005293-A1 5-Membered Heterocyclic Amides And Related Compounds MINDIMMUNE THERAPEUTICS, INC. 2015-01-01 US disclosed
US-20150005293-A1 5-Membered Heterocyclic Amides And Related Compounds MINDIMMUNE THERAPEUTICS, INC. 2015-01-01 US disclosed
US-20150005293-A1 5-Membered Heterocyclic Amides And Related Compounds MINDIMMUNE THERAPEUTICS, INC. 2015-01-01 US disclosed
US-20100292236-A1 5-Membered Heterocyclic Amides And Related Compounds H. LUNDBECK A/S (DK) 2010-11-18 US disclosed
US-20100292236-A1 5-Membered Heterocyclic Amides And Related Compounds H. LUNDBECK A/S (DK) 2010-11-18 US disclosed
US-20100292236-A1 5-Membered Heterocyclic Amides And Related Compounds H. LUNDBECK A/S (DK) 2010-11-18 US disclosed
WO-2009012482-A2 5-MEMBERED HETEROCYCLIC AMIDES AND RELATED COMPOUNDS H.LUNDBECK A/S (DK) 2009-01-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150005293-A1 5-Membered Heterocyclic Amides And Related Compounds GPR35, HCAR2, HCAR1 HPGD 388/4885LMNA 3768/4885SMN1; SMN2 3228/4885
US-20100292236-A1 5-Membered Heterocyclic Amides And Related Compounds GPR35, HCAR2, HCAR1 HPGD 388/4885LMNA 3768/4885SMN1; SMN2 3228/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.