SCHEMBL375054

SCHEMBL375054

C=C(C=Cc1ccccc1)C(=O)Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.57
HDAC3 O15379 2/20 0.57
HDAC4 P56524 2/20 0.57
HDAC1 Q13547 2/20 0.57
HDAC2 Q92769 2/20 0.57
HDAC8 Q9BY41 2/20 0.57
HDAC6 Q9UBN7 2/20 0.57
PLIN1 O60240 2/20 0.57
LMNA P02545 2/20 0.57
RECQL P46063 2/20 0.57
PLIN5 Q00G26 2/20 0.57
ABHD5 Q8WTS1 2/20 0.57
ALDH1A1 P00352 2/20 0.57
F3 P13726 2/20 0.57
CYP1A2 P05177 2/20 0.57
CYP2D6 P10635 2/20 0.57
TNKS O95271 1/20 0.57
HCAR2 Q8TDS4 1/20 0.57
HDAC7 Q8WUI4 1/20 0.57
HDAC10 Q969S8 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7936575 1.00 MAPT (0.57) MAPTHDAC3HDAC4HDAC1HDAC2
SCHEMBL376003 0.83 MAPT (0.61) MAPTHDAC3HDAC4HDAC1HDAC2
SCHEMBL15120 0.83 MAPT (0.61) MAPTHDAC3HDAC4HDAC1HDAC2
SCHEMBL28287153 0.82 MAPT (0.59) MAPTHDAC3HDAC4HDAC1HDAC2
Ammonia Solution, Strong SCHEMBL5175448 0.82 MAPT (0.59) MAPTHDAC3HDAC4HDAC1HDAC2
SCHEMBL16268784 0.82 MAPT (0.59) MAPTHDAC3HDAC4HDAC1HDAC2
SCHEMBL24119310 0.80 GLA (0.64) MAPTHDAC3HDAC4HDAC1HDAC2
Potassium Ion SCHEMBL6578283 0.80 MAPT (0.57) MAPTHDAC3HDAC4HDAC1HDAC2
SCHEMBL3279786 0.80 MAPT (0.57) MAPTHDAC3HDAC4HDAC1HDAC2
SCHEMBL4982120 0.80 MAPT (0.57) MAPTHDAC3HDAC4HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765590-B2 POLYAMIDE-BASED MULTI-LAYER STRUCTURE WHICH IS USED TO COVER SUBSTRATES ARKEMA FRANCE (FR) 2023-03-29 EP disclosed
WO-2012020997-A3 APPARATUS FOR ROTATING A TABLE OF A MACHINING TOOL 두산인프라코어 주식회사 (KR) 2012-05-10 WO disclosed
EP-1765590-B1 POLYAMIDE-BASED MULTI-LAYER STRUCTURE WHICH IS USED TO COVER SUBSTRATES ARKEMA FRANCE (FR) 2012-01-25 EP disclosed
EP-1866370-B1 POLYMER MATERIALS CONTAINING DISPERSED CARBON NANOTUBES ARKEMA FRANCE (FR) 2011-12-07 EP disclosed
EP-1866370-A1 POLYMER MATERIALS CONTAINING DISPERSED CARBON NANOTUBES Arkema France (FR) 2007-12-19 EP disclosed
EP-1725612-A1 THERMOPLASTIC COMPOSITIONS BASED ON OLEFINIC OR STYRENIC POLYMERS AND ALKYL (METH)ACRYLATE COPOLYMERS AND THE THUS OBTAINED LAYERS OR FILMS Arkema France (FR) 2006-11-29 EP disclosed
WO-2006106214-A1 POLYMER MATERIALS CONTAINING DISPERSED CARBON NANOTUBES ARKEMA FRANCE (FR) 2006-10-12 WO disclosed
WO-2005087861-A1 THERMOPLASTIC COMPOSITIONS BASED ON OLEFINIC OR STYRENIC POLYMERS AND ALKYL (METH)ACRYLATE COPOLYMERS AND THE THUS OBTAINED LAYERS OR FILMS ARKEMA FRANCE (FR) 2005-09-22 WO disclosed
EP-1569991-A1 METHOD OF TRAPPING FREE COMPOUNDS CONTAINED IN A POLYMER COMPOSITION CECA S.A. (FR) 2005-09-07 EP disclosed
WO-2004063261-A1 METHOD OF TRAPPING FREE COMPOUNDS CONTAINED IN A POLYMER COMPOSITION CECA S.A. (FR) 2004-07-29 WO disclosed
US-6294593-B1 COMBINING HOST POLYMER WITH GUEST CROSSLINIKING AGENT; EXPOSING COMBINED HOST POLYMER AND GUEST CROSSLINKING AGENT TO ELECTRIC FIELD TO POLE SECOND ORDER NONLINEAR OPTICAL COMPONENT OF POLYMER; EXPOSING TO ELECTROMAGNETIC RADIATION UNIVERSITY OF MASSACHUSETTS LOWELL 2001-09-25 US disclosed