SCHEMBL3754139

SCHEMBL3754139

NC(Cc1ccc(C(F)(F)F)cc1)C1CCCNC1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
KCNH2 Q12809 1/20 0.41
CTSC P53634 1/20 0.40
DPP4 P27487 1/20 0.40
FAP Q12884 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
DPP9 Q86TI2 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
HTR2A P28223 1/20 0.39
HTR2C P28335 2/20 0.38
HTR6 P50406 1/20 0.37
CDK2AP1 O14519 1/20 0.36
CHEK1 O14757 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27602391 0.73 SLC6A2 (0.40) SLC6A2SLC6A4DPP4FAPDPP8
SCHEMBL27644931 0.73 EED (0.48) SLC6A2SLC6A4KCNH2HTR2AHTR2C
SCHEMBL13576641 0.73 EED (0.48) SLC6A2SLC6A4KCNH2HTR2AHTR2C
SCHEMBL27288939 0.72 GBA1 (0.43) SLC6A2SLC6A4DPP4
SCHEMBL5188031 0.72 PNMT (0.48) SLC6A2SLC6A4HTR2C
SCHEMBL8330460 0.71 CTSC (0.46) SLC6A2SLC6A4KCNH2CTSCDPP4
SCHEMBL3662366 0.71 SLC6A2 (0.56) SLC6A2SLC6A4KCNH2HTR2AHTR6
SCHEMBL3444214 0.70 MAOB (0.49) HTR2A
SCHEMBL10435882 0.70 FLT3 (0.39) KCNH2
Hydrochloric Acid SCHEMBL31599129 0.70 SLC6A2 (0.46) SLC6A2SLC6A4CTSCHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170058-A1 CETP INHIBITORS DERIVED FROM BENZOXAZOLE ARYLAMIDES Merck Sharp & Dohme Corp. (US) 2010-04-07 EP disclosed
WO-2008156715-A1 CETP INHIBITORS DERIVED FROM BENZOXAZOLE ARYLAMIDES MERCK & CO., INC. (US) 2008-12-24 WO disclosed