SCHEMBL3662366

SCHEMBL3662366

FC(F)(F)c1ccc(C(c2ccccc2)C2CCCNC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.56
SLC6A4 P31645 1/20 0.56
HTR6 P50406 1/20 0.42
KCNH2 Q12809 1/20 0.41
TACR1 P25103 1/20 0.40
HTR2A P28223 1/20 0.40
ACP3 P15309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649264 0.87 SLC6A2 (0.43) SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL8983761 0.85 SLC6A2 (0.42) SLC6A2SLC6A4
SCHEMBL23848782 0.84 SLC6A2 (0.47) SLC6A2SLC6A4
SCHEMBL3660818 0.82 SLC6A2 (0.58) SLC6A2SLC6A4TACR1ACP3
SCHEMBL25501912 0.81 SLC6A2 (0.44) SLC6A2SLC6A4
SCHEMBL3725941 0.81 SLC6A2 (0.86) SLC6A2SLC6A4
SCHEMBL3719834 0.81 SLC6A2 (0.86) SLC6A2SLC6A4
SCHEMBL3715944 0.81 SLC6A2 (0.86) SLC6A2SLC6A4
SCHEMBL3719829 0.81 SLC6A2 (0.86) SLC6A2SLC6A4
SCHEMBL13152467 0.81 SLC6A2 (0.86) SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230146127-A1 3-DIARYLMETHYLENES AND USES THEREOF ATUX ISKAY LLC 2023-05-11 US disclosed
WO-2021188949-A1 3-DIARYLMETHYLENES AND USES THEREOF ATUX ISKAY LLC (US) 2021-09-23 WO disclosed
US-8258306-B2 Glycine transporter-1 inhibitors AMGEN INC. (US) 2012-09-04 US disclosed
US-20100298341-A1 Glycine Transporter-1 Inhibitors AMGEN INC. 2010-11-25 US disclosed
EP-2231601-A2 GLYCINE TRANSPORTER-1 INHIBITORS Amgen, Inc (US) 2010-09-29 EP disclosed
WO-2009075857-A2 GLYCINE TRANSPORTER-1 INHIBITORS AMGEN INC. (US) 2009-06-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230146127-A1 3-DIARYLMETHYLENES AND USES THEREOF MYC, MYCBP, FOXO1 SLC6A2 4182/4885SLC6A4 4333/4885HTR6 3590/4885
US-20100298341-A1 Glycine Transporter-1 Inhibitors SLC18A2, SLC7A11, SLC6A5 SLC6A2 7/4885SLC6A4 16/4885HTR6 338/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.