SCHEMBL375882

SCHEMBL375882

CC(C)(C)C(Br)C[C@H](NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.56
CTSL P07711 6/20 0.56
CTSB P07858 3/20 0.56
CTSK P43235 9/20 0.54
PPARA Q07869 3/20 0.52
PPARG P37231 1/20 0.52
ITGB3 P05106 2/20 0.52
ITGA2B P08514 2/20 0.52
ALDH1A1 P00352 1/20 0.49
ALOX15 P16050 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27857330 0.86 CTSK (0.55) CTSSCTSLCTSBCTSKPPARA
SCHEMBL2776839 0.86 CTSK (0.55) CTSSCTSLCTSBCTSKPPARA
SCHEMBL42878 0.86 CTSK (0.55) CTSSCTSLCTSBCTSKPPARA
SCHEMBL2366985 0.82 CTSK (0.76) CTSSCTSLCTSBCTSK
SCHEMBL1823902 0.82 CTSK (0.76) CTSSCTSLCTSBCTSK
SCHEMBL222158 0.82 CTSK (0.76) CTSSCTSLCTSBCTSK
SCHEMBL2400096 0.81 CTSS (0.71) CTSSCTSLCTSBCTSKPPARA
SCHEMBL3824323 0.81 CTSS (0.71) CTSSCTSLCTSBCTSKPPARA
SCHEMBL8683808 0.81 CTSK (0.62) CTSSCTSLCTSBCTSK
SCHEMBL7580108 0.81 CTSK (0.62) CTSSCTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079743-B1 PTERIDINE DERIVATIVES AS POLO-LIKE KINASE INHIBITORS USEFUL IN THE TREATMENT OF CANCER CHROMA THERAPEUTICS LTD (GB) 2012-01-25 EP disclosed