SCHEMBL3758935

SCHEMBL3758935

O=C(O)c1ccc(Nc2nc3ccccc3o2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.71
RAB9A P51151 5/20 0.71
SMN1; SMN2 Q16637 3/20 0.71
GAA P10253 2/20 0.71
NPSR1 Q6W5P4 2/20 0.71
ALDH1A1 P00352 1/20 0.71
PKM P14618 1/20 0.71
HDAC6 Q9UBN7 3/20 0.60
SCD O00767 1/20 0.57
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
MAPT P10636 3/20 0.56
ATM Q13315 1/20 0.55
ABCC1 P33527 1/20 0.53
ABCG2 Q9UNQ0 1/20 0.53
SIRT5 Q9NXA8 1/20 0.52
GALK1 P51570 1/20 0.52
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
HPGD P15428 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20458131 0.88 NPC1 (0.67) NPC1RAB9ASMN1; SMN2GAANPSR1
SCHEMBL13058942 0.87 NPC1 (0.65) NPC1RAB9ASMN1; SMN2GAANPSR1
Acetic Acid SCHEMBL7433376 0.85 NPC1 (0.81) NPC1RAB9ASMN1; SMN2GAANPSR1
SCHEMBL11380131 0.85 NPC1 (0.66) NPC1RAB9ASMN1; SMN2GAANPSR1
SCHEMBL2658434 0.84 NPC1 (1.00) NPC1RAB9ASMN1; SMN2GAANPSR1
SCHEMBL31430548 0.84 HDAC6 (0.62) NPC1RAB9ASMN1; SMN2GAANPSR1
SCHEMBL31430584 0.84 NPC1 (0.56) NPC1RAB9ASMN1; SMN2GAANPSR1
SCHEMBL13002091 0.83 NPC1 (0.60) NPC1RAB9ASMN1; SMN2GAANPSR1
SCHEMBL22703575 0.83 NPC1 (0.60) NPC1RAB9ASMN1; SMN2GAANPSR1
SCHEMBL3453070 0.83 ELANE (0.76) NPC1RAB9ASMN1; SMN2NPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8486370-B2 Heterocyclic ligands for integrin imaging and therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-07-16 US disclosed
US-8486370-B2 Heterocyclic ligands for integrin imaging and therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-07-16 US disclosed
US-8486370-B2 Heterocyclic ligands for integrin imaging and therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-07-16 US disclosed
US-20100310455-A1 Heterocyclic Ligands for Integrin Imaging and Therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2010-12-09 US disclosed
US-20100310455-A1 Heterocyclic Ligands for Integrin Imaging and Therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2010-12-09 US disclosed
US-20100310455-A1 Heterocyclic Ligands for Integrin Imaging and Therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2010-12-09 US disclosed
WO-2008031016-A2 HETEROCYCLIC LIGANDS FOR INTEGRIN IMAGING AND THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2008-03-13 WO disclosed
US-4275210-A IMMUNOSUPPRESSIVE AGENTS, ANTIFERTILITY AGENTS, PROPHYLAXIS OF MAREK'S DISEASE IN CHICKENS AND HERBICIDES ELI LILLY AND COMPANY (US) 1981-06-23 US disclosed
US-4088770-A ANTIFERTILITY, HERBICIDES ELI LILLY AND COMPANY (US) 1978-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100310455-A1 Heterocyclic Ligands for Integrin Imaging and Therapy ITGA1, ITGAL, ITGA4 NPC1 3565/4885RAB9A 1592/4885SMN1; SMN2 2082/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.