SCHEMBL3765532

SCHEMBL3765532

CCc1cccc(-c2ccc(N3CCN(CC(=O)N4CCN(C5CCC5)CC4)CC3)nn2)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.44
RAB9A P51151 7/20 0.44
HRH3 Q9Y5N1 2/20 0.41
DRD2 P14416 2/20 0.41
DRD4 P21917 2/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GRIN2B Q13224 4/20 0.40
PAX8 Q06710 2/20 0.40
MEN1 O00255 1/20 0.40
HSP90AA1 P07900 1/20 0.40
KMT2A Q03164 1/20 0.40
TP53 P04637 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3771707 0.89 GRM5 (0.46) NPC1RAB9AHRH3KDM4EHTT
SCHEMBL3767452 0.89 LMNA (0.45) NPC1RAB9AHRH3KDM4EALDH1A1
SCHEMBL3769164 0.89 TP53 (0.45) NPC1RAB9AHRH3HTTNPSR1
SCHEMBL3768006 0.88 NPC1 (0.42) NPC1RAB9AHRH3KDM4EALDH1A1
SCHEMBL3776330 0.88 GRIN2B (0.43) HRH3DRD2DRD4KDM4EALDH1A1
SCHEMBL3770272 0.88 CYP11B1 (0.44) NPC1RAB9AHRH3HTTPAX8
SCHEMBL3774634 0.88 KMT2A (0.49) NPC1RAB9AHRH3KDM4EALDH1A1
SCHEMBL3765840 0.87 TP53 (0.45) NPC1RAB9AHRH3KDM4EALDH1A1
SCHEMBL3773927 0.87 ALDH1A1 (0.47) RAB9AHRH3KDM4EALDH1A1HTT
SCHEMBL3780577 0.87 NPC1 (0.41) NPC1RAB9AHRH3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851474-B2 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION (US) 2010-12-14 US disclosed
US-7851474-B2 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION (US) 2010-12-14 US disclosed
US-20070049571-A1 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION 2007-03-01 US disclosed
US-20070049571-A1 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION 2007-03-01 US disclosed
WO-2007016496-A2 DIPIPERAZINYL KETONES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2007-02-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070049571-A1 Dipiperazinyl ketones and related analogues HRH4, HRH3, HRH1 NPC1 3462/4885RAB9A 3824/4885HRH3 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.