SCHEMBL3765643

SCHEMBL3765643

C=CCN1CNCC1=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL7155879 0.98 CYP3A4 (0.37)
SCHEMBL1754879 0.80 CYP3A4 (0.35)
SCHEMBL979256 0.80 CYP3A4 (0.35)
Hydrochloric Acid SCHEMBL2898888 0.79 CYP3A4 (0.34)
SCHEMBL5342102 0.77 SLC6A2 (0.36)
SCHEMBL9304982 0.75 CYP3A4 (0.38)
SCHEMBL5139880 0.72
SCHEMBL24738965 0.71
SCHEMBL9836861 0.70 CYP3A4 (0.46)
SCHEMBL10696089 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8933276-B2 Heterogeneous chiral catalyst AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-01-13 US claimed
EP-1973656-B1 HETEROGENEOUS CHIRAL CATALYST AGENCY SCIENCE TECH & RES (SG) 2012-05-16 EP claimed
US-20090281358-A1 HETEROGENEOUS CHIRAL CATALYST AGENCY FOR SCIENCE TECHNOLOGY AND RESEARCH (SG) 2009-11-12 US claimed
EP-1973656-A4 HETEROGENEOUS CHIRAL CATALYST AGENCY SCIENCE TECH & RES (SG) 2009-08-05 EP claimed
EP-1973656-A1 HETEROGENEOUS CHIRAL CATALYST Agency for Science, Technology and Research (SG) 2008-10-01 EP claimed
WO-2007084075-A1 HETEROGENEOUS CHIRAL CATALYST AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2007-07-26 WO claimed
US-8933276-B2 Heterogeneous chiral catalyst AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-01-13 US disclosed
EP-1973656-B1 HETEROGENEOUS CHIRAL CATALYST AGENCY SCIENCE TECH & RES (SG) 2012-05-16 EP disclosed
US-20090281358-A1 HETEROGENEOUS CHIRAL CATALYST AGENCY FOR SCIENCE TECHNOLOGY AND RESEARCH (SG) 2009-11-12 US disclosed
EP-1973656-A4 HETEROGENEOUS CHIRAL CATALYST AGENCY SCIENCE TECH & RES (SG) 2009-08-05 EP disclosed
EP-1973656-A1 HETEROGENEOUS CHIRAL CATALYST Agency for Science, Technology and Research (SG) 2008-10-01 EP disclosed
WO-2007084075-A1 HETEROGENEOUS CHIRAL CATALYST AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2007-07-26 WO disclosed
US-3971757-A STABILIZERS FOR POLYMERS CIBA-GEIGY CORPORATION (US) 1976-07-27 US disclosed