SCHEMBL3770495

SCHEMBL3770495

CCOC(=O)OC[C@H]1O[C@@](O)(Oc2nn(C(C)C)c(C)c2Cc2ccc(OC)cc2F)[C@H](O)[C@@H](O)[C@@H]1O

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC5A1 P13866 5/20 0.51
SLC5A2 P31639 5/20 0.51
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
P2RX7 Q99572 1/20 0.30
EED O75530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3771058 0.96 SLC5A1 (0.45) SLC5A1SLC5A2MEN1POLBHTT
SCHEMBL3779489 0.95 SLC5A1 (0.45) SLC5A1SLC5A2MEN1POLBHTT
SCHEMBL3769460 0.94 SLC5A1 (0.51) SLC5A1SLC5A2P2RX7
SCHEMBL3768834 0.94 SLC5A1 (0.58) SLC5A1SLC5A2P2RX7
SCHEMBL3766872 0.93 SLC5A1 (0.42) SLC5A1SLC5A2MEN1POLBHTT
SCHEMBL3773516 0.93 SLC5A1 (0.42) SLC5A1SLC5A2MEN1POLBHTT
SCHEMBL3770840 0.93 SLC5A1 (0.44) SLC5A1SLC5A2
SCHEMBL3768991 0.92 SLC5A1 (0.43) SLC5A1SLC5A2MEN1POLBHTT
SCHEMBL3766867 0.92 SLC5A1 (0.47) SLC5A1SLC5A2P2RX7
SCHEMBL3771132 0.92 SLC5A1 (0.49) SLC5A1SLC5A2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070072813-A1 Methods for preventing and treating metabolic disorders and new pyrazole-O-glycoside derivatives AJINOMOTO CO., INC. (JP) 2007-03-29 US claimed
US-20100317575-A1 PHARMACEUTICAL COMPOSITION COMPRISING A PYRAZOLE-O-GLUCOSIDE DERIVATIVE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-16 US disclosed
US-20070072813-A1 Methods for preventing and treating metabolic disorders and new pyrazole-O-glycoside derivatives AJINOMOTO CO., INC. (JP) 2007-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070072813-A1 Methods for preventing and treating metabolic disorders and new pyrazole-O-glycoside derivatives IAPP, G6PC1, GPR119 SLC5A1 4/4885SLC5A2 6/4885MEN1 2486/4885
US-20100317575-A1 PHARMACEUTICAL COMPOSITION COMPRISING A PYRAZOLE-O-GLUCOSIDE DERIVATIVE SLC5A1, SLC5A2, G6PC1 SLC5A1 1/4885SLC5A2 2/4885MEN1 3761/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.