SCHEMBL377235

SCHEMBL377235

Fc1cc(CBr)c(F)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.39
KDM1B Q8NB78 1/20 0.39
GPR84 Q9NQS5 1/20 0.37
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTR2A P28223 9/20 0.33
HTR2C P28335 8/20 0.33
HTR2B P41595 6/20 0.33
SLC6A4 P31645 1/20 0.33
KCNH2 Q12809 1/20 0.33
DPP4 P27487 1/20 0.32
MAPT P10636 1/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2C9 P11712 2/20 0.31
PLA2G1B P04054 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
ATG4B Q9Y4P1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30474348 1.00 KDM1A (0.39) KDM1AKDM1BGPR84ALDH1A1TDP1
SCHEMBL31266184 0.91 GPR84 (0.37) KDM1AKDM1BGPR84ALDH1A1TDP1
SCHEMBL693457 0.91 GPR84 (0.37) KDM1AKDM1BGPR84ALDH1A1TDP1
SCHEMBL11027502 0.88 GPR84 (0.36) KDM1AKDM1BGPR84ALDH1A1TDP1
SCHEMBL3875287 0.88 GPR84 (0.38) KDM1AKDM1BGPR84ALDH1A1TDP1
SCHEMBL488821 0.86 GPR84 (0.37) KDM1AKDM1BGPR84ALDH1A1TDP1
SCHEMBL18226969 0.84 DPP4 (0.39) DPP4
SCHEMBL14774772 0.83 DPP4 (0.33) KDM1AKDM1BGPR84DPP4MAPT
SCHEMBL30030017 0.83 DPP4 (0.33) KDM1AKDM1BGPR84DPP4MAPT
SCHEMBL3363763 0.82 KDM1A (0.38) KDM1AKDM1BGPR84ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4605394-A1 PYRIMIDINE SGC STIMULATORS Tisento Therapeutics Inc. (US) 2025-08-27 EP disclosed
US-20250223307-A1 MDM2/MDMX DOUBLE-TARGET INHIBITOR COMPOUND, PRODRUG, PHARMACEUTICAL COMPOSITION, AND PREPARATION METHOD THEREFOR AND USE THEREOF GLOBAL HEALTH DRUG DISCOVERY INSTITUTE (CN) 2025-07-10 US disclosed
US-20250122171-A1 Substituted Amine Compounds, Compositions and Methods of Use DEEP APPLE THERAPEUTICS, INC. 2025-04-17 US disclosed
US-20250109148-A1 HETEROCYCLIC GLP-1 AGONISTS SHANGHAI SHOUTI BIOTECHNOLOGY CO., LTD. (CN) 2025-04-03 US disclosed
WO-2024104304-A1 MDM2/MDMX DOUBLE-TARGET INHIBITOR COMPOUND, PRODRUG, PHARMACEUTICAL COMPOSITION, AND PREPARATION METHOD THEREFOR AND USE THEREOF 北京华益健康药物研究中心 2024-05-23 WO disclosed
WO-2024086179-A1 PYRIMIDINE SGC STIMULATORS TISENTO THERAPEUTICS, INC. (US) 2024-04-25 WO disclosed
EP-2408760-A1 THIOPHENYL SULFONAMIDES FOR THE TREATMENT OF ALZHEIMER'S DISEASE Bristol-Myers Squibb Company (US) 2012-01-25 EP disclosed
US-20110071199-A1 Thiophenyl Sulfonamides for the Treatment of Alzheimer's Disease BRISTOL-MYERS SQUIBB COMPANY 2011-03-24 US disclosed
WO-2010107997-A1 THIOPHENYL SULFONAMIDES FOR THE TREATMENT OF ALZHEIMER'S DISEASE BRISTOL-MYERS SQUIBB COMPANY (US) 2010-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250122171-A1 Substituted Amine Compounds, Compositions and Methods of Use MRGPRX2, MRGPRX1, MRGPRX4 KDM1A 4314/4885KDM1B 2900/4885GPR84 357/4885
US-20250109148-A1 HETEROCYCLIC GLP-1 AGONISTS GLP1R, GIPR, GCGR KDM1A 1735/4885KDM1B 2790/4885GPR84 123/4885
US-20110071199-A1 Thiophenyl Sulfonamides for the Treatment of Alzheimer's Disease APP, PSEN1, PSEN2 KDM1A 2970/4885KDM1B 4093/4885GPR84 1415/4885
US-20250223307-A1 MDM2/MDMX DOUBLE-TARGET INHIBITOR COMPOUND, PRODRUG, PHARMACEUTICAL COMPOSITION, AND PREPARATION METHOD THEREFOR AND USE THEREOF MDM2, TP53, TP53BP1 KDM1A 2372/4885KDM1B 2687/4885GPR84 3211/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.