SCHEMBL3774043

SCHEMBL3774043

O=C(C=Cc1ccc(Cl)c(Cl)c1)N1CCN(CC(=O)N2CCN(C3CCC3)CC2)CC1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPR183 P32249 7/20 0.58
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
CCR2 P41597 8/20 0.52
SLC2A1 P11166 1/20 0.46
HRH3 Q9Y5N1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3774031 1.00 GPR183 (0.58) GPR183NPC1RAB9ATDP1CCR2
SCHEMBL3767721 0.89 MEN1 (0.56) GPR183NPC1RAB9ACCR2HRH3
SCHEMBL3767727 0.89 MEN1 (0.56) GPR183NPC1RAB9ACCR2HRH3
SCHEMBL3773067 0.87 MEN1 (0.54) GPR183NPC1HRH3
SCHEMBL3773064 0.87 MEN1 (0.54) GPR183NPC1HRH3
SCHEMBL3765623 0.84 ALDH1A1 (0.58) GPR183HRH3
SCHEMBL3765617 0.84 ALDH1A1 (0.58) GPR183HRH3
SCHEMBL3773866 0.84 MEN1 (0.56) GPR183NPC1RAB9A
SCHEMBL3773864 0.84 MEN1 (0.56) GPR183NPC1RAB9A
SCHEMBL3769147 0.83 TDP1 (0.52) NPC1RAB9ATDP1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851474-B2 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION (US) 2010-12-14 US disclosed
US-7851474-B2 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION (US) 2010-12-14 US disclosed
US-20070049571-A1 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION 2007-03-01 US disclosed
US-20070049571-A1 Dipiperazinyl ketones and related analogues NEUROGEN CORPORATION 2007-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070049571-A1 Dipiperazinyl ketones and related analogues HRH4, HRH3, HRH1 GPR183 59/4885NPC1 3462/4885RAB9A 3824/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.