SCHEMBL377434

SCHEMBL377434

NC1CCN(c2ccc(F)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.59
MAPT P10636 2/20 0.59
MAPK1 P28482 2/20 0.59
LMNA P02545 1/20 0.59
HTT P42858 1/20 0.59
GFER P55789 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
NOTUM Q6P988 1/20 0.50
KDM4E B2RXH2 2/20 0.48
TP53 P04637 2/20 0.48
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
POLB P06746 1/20 0.46
HRH3 Q9Y5N1 1/20 0.45
CA12 O43570 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20495181 0.94 ALDH1A1 (0.53) ALDH1A1MAPTMAPK1LMNAHTT
SCHEMBL1238827 0.88 NOTUM (0.56) ALDH1A1MAPTMAPK1LMNAHTT
SCHEMBL1413520 0.88 NOTUM (0.56) ALDH1A1MAPTMAPK1LMNAHTT
SCHEMBL1413366 0.88 NOTUM (0.56) ALDH1A1MAPTMAPK1LMNAHTT
Hydrochloric Acid SCHEMBL16422372 0.86 NOTUM (0.54) ALDH1A1MAPTMAPK1LMNAHTT
Hydrochloric Acid SCHEMBL16422371 0.86 NOTUM (0.54) ALDH1A1MAPTMAPK1LMNAHTT
Hydrochloric Acid SCHEMBL16422413 0.86 NOTUM (0.54) ALDH1A1MAPTMAPK1LMNAHTT
SCHEMBL22570271 0.82 ALDH1A1 (0.53) ALDH1A1MAPTMAPK1LMNAHTT
SCHEMBL30582885 0.82 ALDH1A1 (0.52) ALDH1A1MAPTMAPK1LMNAHTT
SCHEMBL3441371 0.81 MAPT (0.57) ALDH1A1MAPTMAPK1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 83 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107428730-B 1,3, 5-triazinyl PI3K inhibitors as anti-cancer agents and methods of making the same 科学与工业研究会 2020-10-16 CN claimed
US-20260070884-A1 Inhibitors of Dihydroceramide Desaturase for Treating Disease CENTAURUS THERAPEUTICS (US) 2026-03-12 US disclosed
US-12247019-B2 Inhibitors of dihydroceramide desaturase for treating disease CENTAURUS THERAPEUTICS (US) 2025-03-11 US disclosed
US-20230357187-A1 Inhibitors of Dihydroceramide Desaturase For Treating Disease CENTAURUS THERAPEUTICS 2023-11-09 US disclosed
US-20230357187-A1 Inhibitors of Dihydroceramide Desaturase For Treating Disease CENTAURUS THERAPEUTICS 2023-11-09 US disclosed
US-20230357187-A1 Inhibitors of Dihydroceramide Desaturase For Treating Disease CENTAURUS THERAPEUTICS 2023-11-09 US disclosed
CN-111787916-B Dihydroceramide desaturase inhibitors for treating diseases 森陶鲁斯治疗公司 2023-09-05 CN disclosed
US-11713320-B2 5-heteroaryl substituted indazole-3-carboxamides and preparation and use thereof BIOSPLICE THERAPEUTICS, INC. (US) 2023-08-01 US disclosed
US-11713320-B2 5-heteroaryl substituted indazole-3-carboxamides and preparation and use thereof BIOSPLICE THERAPEUTICS, INC. (US) 2023-08-01 US disclosed
US-11597715-B2 Inhibitors of dihydroceramide desaturase for treating disease CENTAURUS THERAPEUTICS (US) 2023-03-07 US disclosed
US-7183290-B2 Fluoropyrrolidines as dipeptidyl peptidase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 2007-02-27 US disclosed
WO-2007012479-A2 BENZYLPIPERAZINE DERIVATES AND THEIR MEDICAL USE GLAXO GROUP LIMITED (GB) 2007-02-01 WO disclosed
US-20040242636-A1 Enzyme inhibitors as antiinflammatory ageents for psoriasis, obesity SMITHKLINE BEECHAM CORPORATION 2004-12-02 US disclosed
EP-1399433-A2 FLUOROPYRROLIDINES AS DIPEPTIDYL PEPTIDASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-03-24 EP disclosed
WO-2003002553-A2 FLUOROPYRROLIDINES AS DIPEPTIDYL PEPTIDASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-01-09 WO disclosed
US-5723450-A Substituted pyridines, their preparation, and their use as pesticides and fungicides HOECHST SCHERING AGREVO GMBH (DE) 1998-03-03 US disclosed
EP-0719256-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES Hoechst Schering AgrEvo GmbH (DE) 1996-07-03 EP disclosed
WO-1995007891-A1 SUBSTITUTED PYRIDINES, PROCESS FOR PRODUCING THEM AND THEIR USE AS PESTICIDES AND FUNGICIDES HOECHST SCHERING AGREVO GMBH (DE) 1995-03-23 WO disclosed
CN-1080918-A Novel aminopropanol derivatives, pharmaceutical compositions containing them and process for preparing them RICHTER GEDEON VEGYESZET (HU) 1994-01-19 CN disclosed
WO-1993025528-A1 NOVEL AMINOPROPANOL DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME Richter Gedeon Vegyészeti Gyár Rt. (HU) 1993-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11597715-B2 Inhibitors of dihydroceramide desaturase for treating disease CERS2, SMPD1, ASAH1 ALDH1A1 1260/4885MAPT 2085/4885MAPK1 2698/4885
US-20260070884-A1 Inhibitors of Dihydroceramide Desaturase for Treating Disease CERS2, DEGS1, CERT1 ALDH1A1 1500/4885MAPT 4429/4885MAPK1 3314/4885
US-20040242636-A1 Enzyme inhibitors as antiinflammatory ageents for psoriasis, obesity DPP4, DPP7, DPP3 ALDH1A1 531/4885MAPT 2441/4885MAPK1 2837/4885
US-12247019-B2 Inhibitors of dihydroceramide desaturase for treating disease CERS2, SMPD1, ASAH1 ALDH1A1 1260/4885MAPT 2085/4885MAPK1 2698/4885
US-11713320-B2 5-heteroaryl substituted indazole-3-carboxamides and preparation and use thereof DYRK1A, WNT3, DYRK3 ALDH1A1 3709/4885MAPT 201/4885MAPK1 2001/4885
US-20230357187-A1 Inhibitors of Dihydroceramide Desaturase For Treating Disease CERS2, SMPD1, ASAH1 ALDH1A1 1260/4885MAPT 2085/4885MAPK1 2698/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.