SCHEMBL378063

SCHEMBL378063

CC1(C)OB(C2=CCN(C(=O)O)CC2)OC1(C)C

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.46
MAPK1 P28482 1/20 0.44
F2 P00734 1/20 0.32
F11 P03951 1/20 0.32
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
PRSS3 P35030 1/20 0.32
P4HB P07237 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
ROCK1 Q13464 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL986716 0.91 P2RX7 (0.51) P2RX7MAPK1F2F11PRSS1
SCHEMBL29756950 0.89 P2RX7 (0.38) P2RX7MAPK1
SCHEMBL20606348 0.88 P2RX7 (0.54) P2RX7MAPK1P4HBROCK1
SCHEMBL2491645 0.88 P2RX7 (0.46) P2RX7MAPK1ROCK1
SCHEMBL12294233 0.87 P2RX7 (0.45) P2RX7MAPK1
SCHEMBL2037752 0.87 P2RX7 (0.45) P2RX7MAPK1F2F11PRSS1
SCHEMBL27972050 0.86 P2RX7 (0.34) P2RX7MAPK1
SCHEMBL370271 0.84 P2RX7 (0.41) P2RX7MAPK1F2F11PRSS1
SCHEMBL28954013 0.84 P2RX7 (0.43) P2RX7MAPK1ROCK1
SCHEMBL22657130 0.84 P2RX7 (0.43) P2RX7MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 498 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4676922-A1 BIFUNCTIONAL COMPOUNDS CAPABLE OF DEGRADING ANDROGEN RECEPTORS Astrazeneca AB (SE) 2026-01-14 EP disclosed
EP-4321514-B1 COMPOUND HAVING ALK INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF CGENETECH SUZHOU CHINA CO LTD (CN) 2025-12-03 EP disclosed
US-20250288595-A1 TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS GENZYME CORP (US) 2025-09-18 US disclosed
US-12318392-B2 Tropomyosin-related kinase (trk) inhibitors GENZYME CORPORATION (US) 2025-06-03 US disclosed
EP-3778597-B1 TETRAHYDROISOQUINOLINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USES THEREOF SICHUAN KELUN BIOTECH BIOPHARMACEUTICAL CO LTD (CN) 2025-05-28 EP disclosed
WO-2024189488-A1 BIFUNCTIONAL COMPOUNDS CAPABLE OF DEGRADING ANDROGEN RECEPTORS ASTRAZENECA AB (SE) 2024-09-19 WO disclosed
CN-118459485-A Amino-substituted heterocycles for the treatment of cancers with EGFR mutations 纽威伦特公司 2024-08-09 CN disclosed
US-20240246927-A1 COMPOUNDS WITH ALK INHIBITORY ACTIVITY AND PREPARATION METHOD AND USE THEREOF CGENETECH (SUZHOU, CHINA) CO., LTD. (CN) 2024-07-25 US disclosed
US-12037336-B2 Compounds with activity as inhibitors of the epithelial sodium channel (ENaC) Enterprise Therapeutics Limited (GB) 2024-07-16 US disclosed
CN-118344363-A Tricyclic fused ring derivatives and uses thereof 广东东阳光药业股份有限公司 2024-07-16 CN disclosed
WO-2004072025-A2 SUBSTITUTED N-ARYLHETEROCYCLES, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENTS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-08-26 WO disclosed
WO-2004064764-A2 SUBSTITUTED ALKYL AMIDO PIPERIDINES H. LUNDBECK A/S (DK) 2004-08-05 WO disclosed
WO-2004063198-A1 DIAZEPINOINDOLE DERIVATIVES AS KINASE INHIBITORS PFIZER INC. (US) 2004-07-29 WO disclosed
US-20040122001-A1 Pharmaceutical compounds ELI LILLY AND COMPANY 2004-06-24 US disclosed
US-6727264-B1 MELANIN CONCENTRATING HORMONE-1 RECEPTOR ANTAGONISTS; SLEEP, EATING, SEXUAL DISORDERS SYNAPTIC PHARMACEUTICAL CORPORATION 2004-04-27 US disclosed
WO-2004005257-A1 SECONDARY AMINO ANILINIC PIPERIDINES AS MCH1 ANTAGONISTS AND USES THEREOF H. LUNDBECK A/S (DK) 2004-01-15 WO disclosed
US-20030225098-A1 Kinase inhibitors ABBOTT LABORATORIES 2003-12-04 US disclosed
US-20030225060-A1 Acylated piperidine derivatives as melanocortin-4 receptor agonists MERCK SHARP & DOHME CORP. 2003-12-04 US disclosed
US-20030199525-A1 Kinase inhibitors ABBOTT LABORATORIES 2003-10-23 US disclosed
WO-2003080064-A1 KINASE INHIBITORS ABBOTT LABORATORIES (US) 2003-10-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030199525-A1 Kinase inhibitors MAP3K19, MAP3K9, MAP3K1 P2RX7 2913/4885MAPK1 29/4885F2 3912/4885
US-12318392-B2 Tropomyosin-related kinase (trk) inhibitors NTRK1, NGF, NTRK2 P2RX7 3127/4885MAPK1 199/4885F2 3566/4885
US-12037336-B2 Compounds with activity as inhibitors of the epithelial sodium channel (ENaC) SCNN1B, SCNN1A, SCNN1G P2RX7 548/4885MAPK1 1448/4885F2 3565/4885
US-20240246927-A1 COMPOUNDS WITH ALK INHIBITORY ACTIVITY AND PREPARATION METHOD AND USE THEREOF ALK, ACVR1, ALKBH3 P2RX7 3959/4885MAPK1 843/4885F2 4751/4885
US-20030225098-A1 Kinase inhibitors MAP3K19, MAP3K9, MAP3K1 P2RX7 2337/4885MAPK1 26/4885F2 4141/4885
US-20030225060-A1 Acylated piperidine derivatives as melanocortin-4 receptor agonists MC4R, MC5R, MC3R P2RX7 1350/4885MAPK1 2745/4885F2 4812/4885
US-20250288595-A1 TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS NTRK1, NGF, NTRK2 P2RX7 3127/4885MAPK1 199/4885F2 3566/4885
US-20040122001-A1 Pharmaceutical compounds CYP2D6, LPXN, CYP1B1 P2RX7 1346/4885MAPK1 2496/4885F2 324/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.