SCHEMBL3782033

SCHEMBL3782033

CN(Cc1cc(-c2cccnc2F)c(S(=O)(=O)c2cccnc2)s1)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.37
FEN1 P39748 1/20 0.35
PTGER2 P43116 5/20 0.35
TAS2R14 Q9NYV8 1/20 0.34
SLC40A1 Q9NP59 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
CKS1B P61024 2/20 0.33
SKP2 Q13309 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
LMNA P02545 2/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4125901 0.92 NAMPT (0.35) NAMPTFEN1SLC40A1ALDH1A1
SCHEMBL4126978 0.91 NAMPT (0.34) NAMPTFEN1PTGER2TAS2R14SLC40A1
SCHEMBL4117657 0.90 GPBAR1 (0.33) NAMPTGPBAR1
SCHEMBL4130745 0.90 GPBAR1 (0.40) NAMPTPTGER2SLC40A1GPBAR1ALDH1A1
SCHEMBL3649326 0.89 HTR6 (0.39) ALDH1A1
SCHEMBL4126631 0.88 ALDH1A1 (0.41) NAMPTALDH1A1LMNA
SCHEMBL3654891 0.87 ATM (0.34) NAMPTALDH1A1LMNA
SCHEMBL4132659 0.86 NAMPT (0.39) NAMPTPTGER2ALDH1A1CA12CA1
SCHEMBL4125865 0.86 LIMK2 (0.33) NAMPTALDH1A1HPGDCA12CA1
SCHEMBL4126584 0.86 NAMPT (0.37) NAMPTFEN1PTGER2TAS2R14GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed