SCHEMBL3786169

SCHEMBL3786169

O=C(O)Cn1nnc(-c2ncc(Br)s2)n1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
SCD O00767 10/20 0.44
RECQL P46063 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3100343 0.80 SCD (0.47) MEN1KMT2ASCDRECQL
SCHEMBL1236210 0.79 SCD (0.55) MEN1KMT2ASCD
SCHEMBL16495737 0.71 FFAR2 (0.33)
SCHEMBL3715973 0.71 MEN1 (0.56) MEN1KMT2ASCDRECQL
SCHEMBL3712697 0.71 MEN1 (0.56) MEN1KMT2ASCDRECQL
SCHEMBL3233566 0.70 SCD (0.57) MEN1KMT2ASCDRECQL
SCHEMBL4024534 0.69 HPGD (0.76) MEN1KMT2ARECQL
SCHEMBL16872542 0.69 SCD (0.63) SCD
SCHEMBL3222620 0.69 LMNA (0.43) MEN1KMT2ASCDRECQL
Hydrochloric Acid SCHEMBL3791256 0.68 SCD (0.61) SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2398809-B1 NOVEL SPIRO COMPOUNDS USEFUL AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK CANADA INC (CA) 2015-07-08 EP disclosed
EP-2398809-A1 NOVEL SPIRO COMPOUNDS USEFUL AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE Merck Canada Inc. (CA) 2011-12-28 EP disclosed
WO-2010094120-A1 NOVEL SPIRO COMPOUNDS USEFUL AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2010-08-26 WO disclosed