SCHEMBL3786553

SCHEMBL3786553

C=CCN1CC2CCC1(N(Cc1ccc(S(=O)(=O)CCC)cc1)C(=O)O)CC2

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RORC P51449 8/20 0.32
OPRM1 P35372 3/20 0.32
OPRK1 P41145 2/20 0.32
ALDH1A1 P00352 2/20 0.31
LMNA P02545 1/20 0.31
MMP2 P08253 2/20 0.31
MMP13 P45452 2/20 0.31
OPRD1 P41143 1/20 0.30
CHRM5 P08912 1/20 0.30
LSS P48449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4181995 0.83 NPC1 (0.36) OPRM1OPRK1OPRD1
SCHEMBL3786554 0.79 OPRM1 (0.32) OPRM1OPRK1ALDH1A1LMNAOPRD1
SCHEMBL3704054 0.74 SLC6A9 (0.47)
Hydrochloric Acid SCHEMBL3705815 0.72 SLC6A9 (0.35)
SCHEMBL3706848 0.68 SLC6A9 (0.62)
SCHEMBL7895340 0.68 SLC6A9 (0.62)
SCHEMBL3710881 0.66 CNR2 (0.40) OPRM1LMNA
SCHEMBL3710931 0.65 OPRM1 (0.31) OPRM1OPRD1
SCHEMBL4241763 0.65 SLC6A9 (0.34) OPRM1OPRK1OPRD1
SCHEMBL4238324 0.65 SLC6A9 (0.34) OPRM1OPRK1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010087761-A1 2-AZA-BICYCLO[2.2.2]OCTANE COMPOUNDS AND USES THEREOF ASTRAZENECA AB (SE) 2010-08-05 WO disclosed