SCHEMBL378864

SCHEMBL378864

O=C(Cl)N1CCC(C(=O)NCCc2ccc(F)cc2)(c2ccccc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.57
CHRM3 P20309 1/20 0.57
KMT2A Q03164 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
MEN1 O00255 2/20 0.49
HTT P42858 1/20 0.47
OPRL1 P41146 2/20 0.47
EPHX1 P07099 1/20 0.46
EPHX2 P34913 1/20 0.46
PLAAT3 P53816 1/20 0.45
PLAAT5 Q96KN8 1/20 0.45
PLAAT2 Q9NWW9 1/20 0.45
PLAAT4 Q9UL19 1/20 0.45
CCR3 P51677 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2471734 0.85 EPHX2 (0.53) CHRM5CHRM3KMT2ASMN1; SMN2MEN1
SCHEMBL2472649 0.83 CHRM5 (0.52) CHRM5CHRM3KMT2ASMN1; SMN2MEN1
SCHEMBL2517627 0.83 CHRM5 (0.54) CHRM5CHRM3KMT2ASMN1; SMN2MEN1
SCHEMBL2468618 0.83 CHRM5 (0.54) CHRM5CHRM3KMT2ASMN1; SMN2MEN1
SCHEMBL2471543 0.82 PLAAT3 (0.49) CHRM5CHRM3KMT2ASMN1; SMN2MEN1
SCHEMBL2471846 0.81 CHRM5 (0.50) CHRM5CHRM3KMT2AMEN1EPHX2
SCHEMBL2469451 0.81 PLAAT3 (0.49) CHRM5CHRM3KMT2ASMN1; SMN2MEN1
SCHEMBL378386 0.81 TACR1 (0.57) CHRM5CHRM3KMT2ASMN1; SMN2MEN1
SCHEMBL2473234 0.81 CHRM5 (0.70) CHRM5CHRM3KMT2ASMN1; SMN2MEN1
SCHEMBL14327377 0.81 PLAAT3 (0.48) CHRM5CHRM3KMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408745-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-01-25 EP disclosed
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed