SCHEMBL378386

SCHEMBL378386

O=C(NCCc1ccc(F)cc1)C1(c2ccccc2)CCNCC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.57
CHRM5 P08912 1/20 0.53
CHRM3 P20309 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.51
HTT P42858 1/20 0.51
PLAAT3 P53816 1/20 0.49
PLAAT5 Q96KN8 1/20 0.49
PLAAT2 Q9NWW9 1/20 0.49
PLAAT4 Q9UL19 1/20 0.49
RAB9A P51151 3/20 0.49
NPC1 O15118 2/20 0.49
HDAC1 Q13547 1/20 0.46
OPRM1 P35372 1/20 0.46
POLB P06746 1/20 0.45
LTA4H P09960 1/20 0.45
EPHX2 P34913 1/20 0.45
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL378420 0.94 TACR1 (0.48) TACR1CHRM5CHRM3SMN1; SMN2PLAAT3
SCHEMBL378738 0.92 TACR1 (0.58) TACR1CHRM5CHRM3SMN1; SMN2HTT
SCHEMBL10254952 0.87 TACR1 (0.69) TACR1SMN1; SMN2HTTRAB9ANPC1
SCHEMBL378422 0.85 TACR1 (0.56) TACR1CHRM5CHRM3SMN1; SMN2HTT
SCHEMBL2467338 0.84 CHRM5 (0.74) TACR1CHRM5CHRM3SMN1; SMN2PLAAT3
SCHEMBL378864 0.81 CHRM5 (0.57) CHRM5CHRM3SMN1; SMN2HTTPLAAT3
SCHEMBL6375805 0.80 SMN1; SMN2 (0.57) TACR1CHRM5CHRM3SMN1; SMN2HTT
SCHEMBL476243 0.79 TACR1 (0.71) TACR1SMN1; SMN2HTTHDAC1OPRM1
SCHEMBL6543304 0.78 OPRM1 (0.56) TACR1CHRM5CHRM3SMN1; SMN2HTT
SCHEMBL19273223 0.77 OPRL1 (0.60) TACR1SMN1; SMN2HTTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408745-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-01-25 EP disclosed
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed