SCHEMBL3789573

SCHEMBL3789573

Cc1cccc(NC(=O)c2ccc(N3CCCCC3)nc2)n1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.61
NPC1 O15118 5/20 0.59
RAB9A P51151 4/20 0.59
MAPT P10636 3/20 0.59
LMNA P02545 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
ALDH1A1 P00352 2/20 0.59
HPGD P15428 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
CHRNA7 P36544 3/20 0.56
CHRNA10 Q9GZZ6 3/20 0.56
CHRNA9 Q9UGM1 3/20 0.56
CHRNB2 P17787 1/20 0.54
CHRNB4 P30926 1/20 0.54
CHRNA3 P32297 1/20 0.54
CHRNA4 P43681 1/20 0.54
GRM5 P41594 1/20 0.52
TP53 P04637 1/20 0.51
PKM P14618 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3809249 0.90 KMT2A (0.56) KMT2ANPC1RAB9AMAPTLMNA
SCHEMBL3788680 0.90 KMT2A (0.60) KMT2ARAB9ASMN1; SMN2L3MBTL1CHRNA7
SCHEMBL3782446 0.87 KMT2A (0.57) KMT2ANPC1RAB9AMAPTLMNA
SCHEMBL3782560 0.83 KMT2A (0.55) KMT2ANPC1RAB9ACHRNA7CHRNA10
SCHEMBL2865126 0.81 RAB9A (0.60) KMT2ANPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL3785591 0.78 MAP3K5 (0.51) KMT2ACHRNA7CHRNA10CHRNA9GRM5
SCHEMBL27696834 0.78 MCHR1 (0.60) KMT2ANPC1RAB9AMAPTLMNA
SCHEMBL13296220 0.76 GRM5 (0.82) KMT2ANPC1RAB9AMAPTLMNA
SCHEMBL3787990 0.76 KMT2A (1.00) KMT2ANPC1RAB9AMAPTLMNA
SCHEMBL30175325 0.76 UBE2T (0.56) KMT2ANPC1RAB9ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010143803-A2 NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2010-12-16 WO claimed
WO-2010143803-A2 NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2010-12-16 WO disclosed
WO-2010143803-A2 NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2010-12-16 WO disclosed