SCHEMBL3791950

SCHEMBL3791950

O=C(NCc1ccccc1OC(F)(F)F)c1ccc2nn(C3CCOCC3)c(=O)n2c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.47
ROCK1 Q13464 1/20 0.45
EPHX2 P34913 13/20 0.45
PPARG P37231 2/20 0.43
DDR1 Q08345 1/20 0.42
CYP2C9 P11712 3/20 0.42
CYP2J2 P51589 3/20 0.42
RIPK1 Q13546 1/20 0.42
HSD17B13 Q7Z5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3794531 0.90 ROCK2 (0.47) ROCK2ROCK1EPHX2PPARGCYP2C9
SCHEMBL3786977 0.89 EPHX2 (0.47) ROCK2ROCK1EPHX2DDR1
SCHEMBL3808163 0.87 DDR1 (0.45) ROCK2ROCK1EPHX2DDR1
SCHEMBL3795177 0.86 DDR1 (0.43) ROCK2ROCK1EPHX2DDR1
SCHEMBL3785014 0.86 DDR1 (0.46) DDR1
SCHEMBL13257972 0.85 ROCK2 (0.42) ROCK2ROCK1
SCHEMBL13258575 0.83 DDR1 (0.41) ROCK2ROCK1EPHX2DDR1
SCHEMBL13258576 0.83 DDR1 (0.41) ROCK2ROCK1EPHX2DDR1
SCHEMBL3792501 0.82 CNR2 (0.48) ROCK2ROCK1EPHX2PPARGRIPK1
SCHEMBL3794154 0.82 EPHX2 (0.52) ROCK2ROCK1EPHX2PPARGRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed