SCHEMBL379205

SCHEMBL379205

C#CCC(CC#C)C(=O)O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 5/20 0.64
GRIK2 Q13002 5/20 0.64
HDAC1 Q13547 2/20 0.38
HDAC2 Q92769 2/20 0.38
CHRM1 P11229 1/20 0.38
AKR1A1 P14550 1/20 0.38
CHRM3 P20309 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
ADRA1A P35348 1/20 0.38
HRH1 P35367 1/20 0.38
DRD3 P35462 1/20 0.38
SLC6A3 Q01959 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
SLC1A1 P43005 2/20 0.35
SLC1A2 P43004 2/20 0.35
SLC1A3 P43003 1/20 0.35
TBXAS1 P24557 1/20 0.35
FOLH1 Q04609 2/20 0.33
CYP1A2 P05177 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870462 0.87
SCHEMBL28591034 0.85
SCHEMBL3104177 0.85
SCHEMBL5053789 0.81 CHRM1 (0.62) GRIK1GRIK2HDAC1HDAC2CHRM1
SCHEMBL7557794 0.81 CHRM1 (0.62) GRIK1GRIK2HDAC1HDAC2CHRM1
SCHEMBL7550179 0.81 GRIK1 (0.62) GRIK1GRIK2HDAC1HDAC2CHRM1
SCHEMBL8847145 0.81 GRIK1 (0.52) GRIK1GRIK2HDAC1HDAC2CHRM1
SCHEMBL28435149 0.81 FOLH1 (0.56) GRIK1GRIK2FOLH1CYP2D6MAPT
SCHEMBL8847127 0.79 GRIK1 (0.50) GRIK1GRIK2HDAC1HDAC2CHRM1
SCHEMBL15310777 0.79 GRIK1 (1.00) GRIK1GRIK2SLC1A1SLC1A2SLC1A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117986716-B Medium-high voltage special cable material and preparation method thereof 南方珠江科技有限公司 2024-06-25 CN claimed
CN-117986716-A Medium-high voltage special cable material and preparation method thereof 南方珠江科技有限公司 2024-05-07 CN claimed
CN-104910328-B Fluorine-containing high dielectric property polynorbornene class-poly-(1,6-heptadiyne) based block copolymer and preparation method thereof 华东师范大学 2017-01-04 CN claimed
CN-104403103-B Hyperbranched poly triazole hb-PTA-OEG and its preparation method and application 华东师范大学 2016-06-29 CN claimed
CN-105085756-A Conjugated polyacetylene containing perylene bisimide and preparation method thereof UNIV EAST CHINA NORMAL 2015-11-25 CN claimed
CN-104910328-A Fluorine-containing high-dielectricity polynorbornene-poly(1,6-heptadiyne) block copolymer and preparation method thereof UNIV EAST CHINA NORMAL 2015-09-16 CN claimed
CN-104403103-A Hyperbranched polytriazole hb-PTA-OEG, and preparation method and application thereof UNIV EAST CHINA NORMAL 2015-03-11 CN claimed
US-12503553-B2 Biodegradable drug-polymer conjugate POLYACTIVA PTY LTD (AU) 2025-12-23 US disclosed
US-20240247106-A1 BIODEGRADABLE DRUG-POLYMER CONJUGATE POLYACTIVA PTY LTD (AU) 2024-07-25 US disclosed
EP-2964224-B1 POLYMER CONJUGATE FOR DELIVERY OF A BIOACTIVE AGENT POLYACTIVA PTY LTD (AU) 2024-07-03 EP disclosed
EP-2964224-B1 POLYMER CONJUGATE FOR DELIVERY OF A BIOACTIVE AGENT POLYACTIVA PTY LTD (AU) 2024-07-03 EP disclosed
CN-117986716-B Medium-high voltage special cable material and preparation method thereof 南方珠江科技有限公司 2024-06-25 CN disclosed
CN-117986716-A Medium-high voltage special cable material and preparation method thereof 南方珠江科技有限公司 2024-05-07 CN disclosed
US-20100029888-A1 Click-Reaction Crosslinkable Multicomponent Silicone Compositions WACKER CHEMIE AG (DE) 2010-02-04 US disclosed
CN-1166622-C 2-amino-1, 2-indanes as selective dopamine D3 ligands �������Ŷ���Լ��������˾ 2004-09-15 CN disclosed
EP-0807101-B1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS UPJOHN CO (US) 2001-06-13 EP disclosed
US-5936000-A 2-aminoindans as selective dopamine D3 ligands PHARMACIA & UPJOHN COMPANY (US) 1999-08-10 US disclosed
CN-1172469-A 2 -aminoindans as selective dopamine D3 ligands UPJOHN CO (US) 1998-02-04 CN disclosed
EP-0807101-A1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1997-11-19 EP disclosed
WO-1996023760-A1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1996-08-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240247106-A1 BIODEGRADABLE DRUG-POLYMER CONJUGATE ADRB3, PTGER3, CHRNE GRIK1 1826/4885GRIK2 2332/4885HDAC1 1701/4885
US-12503553-B2 Biodegradable drug-polymer conjugate ADRB3, PTGER3, CHRNE GRIK1 1826/4885GRIK2 2332/4885HDAC1 1701/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.