SCHEMBL3793402

SCHEMBL3793402

O=S(=O)(c1cccc(N2C=CC=C(c3ccnn3-c3ccccc3)N2)c1)c1nc2ccccc2[nH]1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
CYP2C9 P11712 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
NPSR1 Q6W5P4 1/20 0.31
NOD1 Q9Y239 1/20 0.31
TP53 P04637 1/20 0.31
NT5E P21589 1/20 0.30
MAPT P10636 1/20 0.30
PLAUR Q03405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3788606 0.79 MYC (0.35) ALDH1A1TP53NT5EPLAUR
SCHEMBL519309 0.75 PDE10A (0.53) ALDH1A1MAPK1HSD17B10L3MBTL1CYP2C9
SCHEMBL7591549 0.68 L3MBTL1 (0.64) ALDH1A1MAPK1HSD17B10L3MBTL1MMP2
SCHEMBL31448310 0.68 L3MBTL1 (0.64) ALDH1A1MAPK1HSD17B10L3MBTL1MMP2
SCHEMBL27963536 0.65 PDE10A (0.46) ALDH1A1NPSR1NT5E
SCHEMBL3793536 0.64 MAPT (0.43) L3MBTL1TP53NT5EMAPT
SCHEMBL3788317 0.63 NPBWR1 (0.45) ALDH1A1HSD17B10CYP2C9NPSR1NT5E
SCHEMBL22494203 0.62 L3MBTL1 (0.72) ALDH1A1MAPK1HSD17B10L3MBTL1NPSR1
SCHEMBL2496328 0.61 KDM4E (0.34) ALDH1A1NT5EMAPT
SCHEMBL27963560 0.61 PDE10A (0.46) ALDH1A1NPSR1NT5EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393360-A1 PYRIDAZINONE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2011-12-14 EP disclosed
WO-2010090737-A1 PYRIDAZINONE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-12 WO disclosed