SCHEMBL379341

SCHEMBL379341

COc1ccc2c(c1)CCNC2=O

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.67
PARP10 Q53GL7 9/20 0.63
PARP11 Q9NR21 9/20 0.63
RYR2 Q92736 1/20 0.54
PARP1 P09874 2/20 0.51
PDPK1 O15530 1/20 0.51
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
HPGD P15428 1/20 0.50
MTNR1A P48039 1/20 0.50
MTNR1B P49286 1/20 0.50
MAPKAPK2 P49137 1/20 0.49
METAP1 P53582 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323443 1.00 GRM5 (0.67) GRM5PARP10PARP11RYR2PARP1
SCHEMBL3692167 0.90 GRM5 (0.56) GRM5PARP10PARP11RYR2PARP1
SCHEMBL8161680 0.88 PARP11 (0.68) GRM5PARP10PARP11PARP1PDPK1
SCHEMBL29438649 0.87 PARP10 (0.63) GRM5PARP10PARP11RYR2PARP1
SCHEMBL246378 0.87 PARP10 (0.63) GRM5PARP10PARP11RYR2PARP1
SCHEMBL12230826 0.86 PARP10 (0.56) GRM5PARP10PARP11RYR2PARP1
SCHEMBL8154135 0.84 PARP10 (0.69) GRM5PARP10PARP11PARP1PDPK1
SCHEMBL504342 0.84 GRM5 (0.79) GRM5PARP10PARP11MAPKAPK2
SCHEMBL12077584 0.84 RYR2 (0.51) GRM5PARP10PARP11RYR2KDM4E
SCHEMBL21040262 0.83 PARP11 (0.55) GRM5PARP10PARP11PARP1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 332 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12617811-B2 HPK1 inhibitors and uses thereof REGOR PHARMACEUTICALS, INC. (US) 2026-05-05 US disclosed
US-12612424-B2 HPK1 inhibitors and uses thereof REGOR PHARMACEUTICALS, INC. (US) 2026-04-28 US disclosed
US-12577267-B2 Pyrimidine compounds for use as MAP4K1 inhibitors GLENMARK SPECIALITY S.A. (CH) 2026-03-17 US disclosed
CN-121449553-A Synthesis method of 6- (methoxy) -3, 4-dihydro-1 (2H) -isoquinolone 凯美克(上海)医药科技有限公司 2026-02-03 CN disclosed
CN-121449553-A Synthesis method of 6- (methoxy) -3, 4-dihydro-1 (2H) -isoquinolone 凯美克(上海)医药科技有限公司 2026-02-03 CN disclosed
EP-4678644-A1 SUBSTITUTED DIHYDROTHIENOPYRIMIDINE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF Shanghai Yidi Biotechnology Co., Ltd. (CN) 2026-01-14 EP disclosed
CN-114621207-B Compound serving as thyroid hormone beta receptor agonist and application thereof 广东东阳光药业股份有限公司 2025-02-11 CN disclosed
CN-114555585-B HPK1 inhibitors and uses thereof 锐格药业公司 2025-02-11 CN disclosed
CN-114195764-B Compound serving as thyroid hormone beta receptor agonist and application thereof 广东东阳光药业股份有限公司 2025-01-17 CN disclosed
CN-116096370-B HPK1 inhibitors and uses thereof 锐格药业公司 2024-12-20 CN disclosed
EP-0526402-B1 Heteroaryl substituted hydroxylamine derivatives as lipoxygenase inhibitors CIBA GEIGY AG (CH) 1998-01-21 EP disclosed
US-5707994-A USEFUL AS A PLATELET AGGREGATION INHIBITOR, CANCER METASTASIS INHIBITOR, WOUND HEALING AGENT OR A BONE RESORPTION INHIBITOR SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1998-01-13 US disclosed
WO-1997024124-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed
WO-1997024122-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed
CN-1138322-A 2,3-diaminopropionic acid derivative SUMITOMO PHARMA (JP) 1996-12-18 CN disclosed
EP-0725059-A1 2,3-DIAMINOPROPIONIC ACID DERIVATIVE SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1996-08-07 EP disclosed
US-5350761-A Lipoxygenase inhibitors as antiinflammatory agents and antiallergens CIBA-GEIGY CORPORATION (US) 1994-09-27 US disclosed
US-5334600-A Lipoxygenase inhibitors CIBA-GEIGY CORPORATION (US) 1994-08-02 US disclosed
US-5260316-A Lipoxygenase inhibitor CIBA-GEIGY CORPORATION (US) 1993-11-09 US disclosed
EP-0526402-A1 Heteroaryl substituted hydroxylamine derivatives as lipoxygenase inhibitors CIBA-GEIGY AG (CH) 1993-02-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12612424-B2 HPK1 inhibitors and uses thereof NEK11, NEK1, CSNK1A1 GRM5 2942/4885PARP10 810/4885PARP11 604/4885
US-12617811-B2 HPK1 inhibitors and uses thereof MAP2K4, MAP2K1, MAP2K3 GRM5 4700/4885PARP10 1083/4885PARP11 1218/4885
US-12577267-B2 Pyrimidine compounds for use as MAP4K1 inhibitors PTK2B, MAP3K10, MAP3K20 GRM5 4066/4885PARP10 700/4885PARP11 1172/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.