SCHEMBL3795385

SCHEMBL3795385

Fc1cccc(Cl)c1-c1nc(-c2cnc(-c3cc4ccccc4[nH]3)nc2)c[nH]1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGES O14684 16/20 0.40
JAK2 O60674 1/20 0.38
ORAI1 Q96D31 2/20 0.38
CYP2C9 P11712 3/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37
CASP3 P42574 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3799806 0.89 PTGES (0.44) PTGESJAK2ORAI1CYP2C9KDM4E
SCHEMBL3802996 0.82 PTGES (0.43) PTGESJAK2NPC1RAB9A
SCHEMBL3796002 0.79 PTGES (0.43) PTGESJAK2ORAI1
SCHEMBL3794879 0.77 PTGES (0.47) PTGESJAK2ORAI1
SCHEMBL3795117 0.77 PTGES (0.54) PTGESJAK2ORAI1CYP2C9KDM4E
SCHEMBL3796320 0.74 PTGES (0.49) PTGESJAK2ORAI1CYP2C9
SCHEMBL29662800 0.73 PTGES (0.43) PTGESJAK2CYP2C9
SCHEMBL13076361 0.73 PTGES (0.53) PTGESJAK2
SCHEMBL13076230 0.73 PTGES (0.43) PTGESJAK2CYP2C9
SCHEMBL3801417 0.70 PTGES (0.48) PTGESJAK2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed