SCHEMBL3796752

SCHEMBL3796752

Fc1cccc(Cl)c1-c1nc(-c2cc3cc(C#Cc4ccccc4)ccc3o2)c(Br)[nH]1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGES O14684 19/20 0.62
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
PIM1 P11309 1/20 0.43
CSNK2A2 P19784 1/20 0.43
CSNK2B P67870 1/20 0.43
PIM3 Q86V86 1/20 0.43
PIM2 Q9P1W9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3755228 0.84 PTGES (0.57) PTGESPTGS1PTGS2PIM1CSNK2A2
SCHEMBL3796208 0.82 PTGES (0.48) PTGESPTGS1PTGS2
SCHEMBL3790511 0.78 PTGES (0.78) PTGESPTGS1PTGS2
SCHEMBL3795330 0.77 PTGES (1.00) PTGES
SCHEMBL3801179 0.70 PTGES (0.66) PTGESPTGS1PIM1CSNK2A2CSNK2B
SCHEMBL3795969 0.69 PTGES (0.56) PTGESPIM1CSNK2A2CSNK2BPIM3
SCHEMBL12479262 0.69 PTGES (0.75) PTGESPTGS1PTGS2
SCHEMBL3791995 0.68 PTGES (0.53) PTGES
SCHEMBL13075956 0.68 PTGES (0.53) PTGES
SCHEMBL3800146 0.68 PIM1 (0.49) PTGESPIM1CSNK2A2CSNK2BPIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed