SCHEMBL3796208

SCHEMBL3796208

Fc1cccc(Cl)c1-c1nc(-c2cc3cc(C#Cc4ccccc4)ccc3o2)c[nH]1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGES O14684 20/20 0.48
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3795502 0.85 PTGES (0.43) PTGESPTGS1
SCHEMBL3796734 0.85 PTGES (0.43) PTGESPTGS1
SCHEMBL3800146 0.83 PIM1 (0.49) PTGES
SCHEMBL3796752 0.82 PTGES (0.62) PTGESPTGS1PTGS2
SCHEMBL3792228 0.81 PTGES (0.39) PTGES
SCHEMBL3802320 0.78 PTGES (0.40) PTGESPTGS1
SCHEMBL3791130 0.77 PTGES (0.42) PTGESPTGS1
SCHEMBL3790901 0.76 PTGES (0.39) PTGES
SCHEMBL3796674 0.76 PTGES (0.67) PTGES
SCHEMBL3803252 0.76 MAPT (0.39) PTGESPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed