Fenoprofen

Fenoprofen

SCHEMBL3797

CC(C(=O)O)c1cccc(Oc2ccccc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGS1PTGS2

The experimentally established mechanism targets of Fenoprofen. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 known ✓ P23219 5/20 1.00
PTGS2 known ✓ P35354 5/20 0.58
MEN1 O00255 1/20 0.72
CYP2D6 P10635 1/20 0.72
KMT2A Q03164 1/20 0.72
ALOX5 P09917 1/20 0.60
FFAR1 O14842 1/20 0.59
MAPT P10636 2/20 0.58
CXCR1 P25024 2/20 0.58
CXCR2 P25025 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
SLC22A6 Q4U2R8 2/20 0.58
RECQL P46063 1/20 0.58
KDM4E B2RXH2 1/20 0.58
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58
CYP3A4 P08684 1/20 0.58
HPGD P15428 1/20 0.58
MAPK1 P28482 1/20 0.58
PMP22 Q01453 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(S)-Fenoprofen SCHEMBL4492279 1.00 PTGS1 (1.00) PTGS1MEN1CYP2D6KMT2AALOX5
Fenoprofen SCHEMBL11336376 1.00 PTGS1 (1.00) PTGS1MEN1CYP2D6KMT2AALOX5
R-Fenoprofen SCHEMBL4082 1.00 PTGS1 (1.00) PTGS1MEN1CYP2D6KMT2AALOX5
Fenoprofen SCHEMBL29481372 1.00 PTGS1 (1.00) PTGS1MEN1CYP2D6KMT2AALOX5
R-Fenoprofen SCHEMBL30910976 1.00 PTGS1 (1.00) PTGS1MEN1CYP2D6KMT2AALOX5
Fenoprofen SCHEMBL8754928 1.00 PTGS1 (1.00) PTGS1MEN1CYP2D6KMT2AALOX5
Fenoprofen SCHEMBL4081 0.98 PTGS1 (0.97) PTGS1MEN1CYP2D6KMT2AALOX5
Fenoprofen SCHEMBL8706502 0.98 PTGS1 (0.97) PTGS1MEN1CYP2D6KMT2AALOX5
Fenoprofen SCHEMBL11125651 0.98 PTGS1 (0.97) PTGS1MEN1CYP2D6KMT2AALOX5
Fenoprofen SCHEMBL5108677 0.97 PTGS1 (0.94) PTGS1MEN1CYP2D6KMT2AALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 60532 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106917-A1 EDIBLE TRANSMUCOSAL DRUG DELIVERY METHOD USING AN INTERMEDIATE CAPSULE AS A TEMPORARY VESSEL BioPhysics Pharma, Inc. (US) 2026-05-21 WO claimed
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP claimed
EP-4745155-A1 POWDER CONTAINING PARTICLES OF GELATIN DERIVATIVE AND APPLICATION OF SAME IN MEDICAL TREATMENT National Institute for Materials Science (JP) 2026-05-20 EP claimed
US-20260130928-A1 COMBINATION OF AKR1C3 ACTIVATED ANTICANCER PRODRUG COMPOUND AND ANALGESIC DRUG FOR TREATING CANCER PATIENTS ACCOMPANIED BY PAIN ASCENTAWITS PHARMACEUTICALS LTD (CN) 2026-05-14 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-20260115186-A1 PIPERIDINE UREA DERIVATIVES FOR CANCER THERAPY NEUROPN THERAPEUTICS INC. (US) 2026-04-30 US claimed
US-20260115209-A1 COMBINATION THERAPY INCLUDING COX-2 INHIBITOR FOR THE TREATMENT OF CANCER UNIV CALIFORNIA (US) 2026-04-30 US claimed
US-12605345-B2 Transdermal drug delivery system BioPhysics Pharma, Inc. (US) 2026-04-21 US claimed
US-12605432-B2 Combinations for antigen based therapy DIAMYD MEDICAL AB (SE) 2026-04-21 US claimed
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP claimed
US-4282214-A PHOSPHONATES THE PROCTER & GAMBLE COMPANY (US) 1981-08-04 US claimed
US-4279926-A PHENYL ALKANOIC ACID SALT OF AN AMINO ACID SPA-SOCIETA PRODOTTI ANTIBIOTICI S.P.A. (IT) 1981-07-21 US claimed
US-4256108-A Microporous-semipermeable laminated osmotic system ALZA CORPORATION (US) 1981-03-17 US claimed
US-4233314-A X-METHYL-3-PHENOXYBENZENE ACETIC ACID AND ACETAMINOPHEN MCNEILAB, INC. (US) 1980-11-11 US claimed
EP-0012621-A1 Analgesic composition comprising acetaminophen as a potentiating agent McNeilab, Inc. (US) 1980-06-25 EP claimed
US-4208414-A Vinblastine in rheumatoid arthritis ELI LILLY AND COMPANY (US) 1980-06-17 US claimed
US-4185100-A CORTICOSTEROID AND A HYDROTROPIC ACID DERIVATIVE, ENZYME INHIBITORS JOHNSON & JOHNSON (US) 1980-01-22 US claimed
US-4163783-A ACID AND A BIS/2-PYRIDYL-1-OXIDE/DISULFIDE KLEIN ROBERT W 1979-08-07 US claimed
US-4152430-A ANTIINFLAMMATORY AGENTS WILLIAM H. RORER, INC. (US) 1979-05-01 US claimed
US-3985779-A ANTIINFLAMMATORY AND ANALGESIC ACTIVITIES EISAI CO., LTD. (JA) 1976-10-12 US claimed