SCHEMBL3797105

SCHEMBL3797105

N=C(NO)c1ccc(-c2cnc(-c3c(F)cccc3Cl)[nH]2)cn1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGES O14684 10/20 0.55
JAK2 O60674 2/20 0.45
ORAI1 Q96D31 2/20 0.35
GCGR P47871 1/20 0.35
SCN2A Q99250 2/20 0.34
HPGDS O60760 3/20 0.34
NQO2 P16083 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3792008 0.83 PTGES (0.62) PTGESJAK2GCGRSCN2AHPGDS
SCHEMBL3799056 0.82 PTGES (0.40) PTGESJAK2ORAI1GCGR
SCHEMBL3794463 0.81 PTGES (0.67) PTGESJAK2ORAI1SCN2AHPGDS
SCHEMBL3802423 0.81 PTGES (0.57) PTGESJAK2GCGR
SCHEMBL3800707 0.81 PTGES (0.60) PTGESJAK2GCGR
SCHEMBL3796557 0.80 PTGES (0.53) PTGESJAK2GCGR
SCHEMBL3790890 0.79 PTGES (0.53) PTGESJAK2GCGR
SCHEMBL3795105 0.79 PTGES (0.52) PTGESJAK2ORAI1GCGR
SCHEMBL3797910 0.77 PTGES (0.50) PTGESJAK2ORAI1GCGRSCN2A
SCHEMBL3796421 0.76 PTGES (0.54) PTGESJAK2GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed